SCHEMBL3170290

SCHEMBL3170290

CC(C)(O)CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.52
CHRM2 P08172 3/20 0.51
CA12 O43570 1/20 0.50
CA9 Q16790 1/20 0.50
MEN1 O00255 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13484325 0.88 ALDH1A1 (0.52) ALDH1A1CHRM2CA12CA9MEN1
SCHEMBL2372406 0.85 CHRM2 (0.47) ALDH1A1CHRM2CA12CA9MEN1
SCHEMBL5962347 0.83 CHRM2 (0.54) ALDH1A1CHRM2CA12CA9MEN1
SCHEMBL9625482 0.83 CHRM2 (0.63) ALDH1A1CHRM2MEN1CYP1A2CYP2C19
SCHEMBL11681175 0.82 CHRM2 (0.47) ALDH1A1CHRM2CA12CA9MEN1
SCHEMBL7286379 0.82 CHRM2 (0.53) ALDH1A1CHRM2CA12CA9MEN1
SCHEMBL3727196 0.81 CHRM2 (0.56) ALDH1A1CHRM2CA12CA9
SCHEMBL30214381 0.80 CHRM2 (0.51) ALDH1A1CHRM2CA12CA9MEN1
SCHEMBL28964583 0.80 CHRM2 (0.51) ALDH1A1CHRM2CA12CA9MEN1
SCHEMBL5681593 0.80 CHRM2 (0.51) ALDH1A1CHRM2CA12CA9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8703987-B2 Methods for preparing 2-methoxyisobutylisonitrile and tetrakis(2-methoxyisobutylisonitrile)copper(I) tetrafluoroborate Draximage Limited (IE) 2014-04-22 US disclosed
US-8703987-B2 Methods for preparing 2-methoxyisobutylisonitrile and tetrakis(2-methoxyisobutylisonitrile)copper(I) tetrafluoroborate Draximage Limited (IE) 2014-04-22 US disclosed
US-8703987-B2 Methods for preparing 2-methoxyisobutylisonitrile and tetrakis(2-methoxyisobutylisonitrile)copper(I) tetrafluoroborate Draximage Limited (IE) 2014-04-22 US disclosed
US-20100010250-A1 METHODS FOR PREPARING 2-METHOXYISOBUTYLISONITRILE AND TETRAKIS(2-METHOXYISOBUTYLISONITRILE)COPPER(I) TETRAFLUOROBORATE Draximage Limited (IE) 2010-01-14 US disclosed
US-20100010250-A1 METHODS FOR PREPARING 2-METHOXYISOBUTYLISONITRILE AND TETRAKIS(2-METHOXYISOBUTYLISONITRILE)COPPER(I) TETRAFLUOROBORATE Draximage Limited (IE) 2010-01-14 US disclosed
US-20100010250-A1 METHODS FOR PREPARING 2-METHOXYISOBUTYLISONITRILE AND TETRAKIS(2-METHOXYISOBUTYLISONITRILE)COPPER(I) TETRAFLUOROBORATE Draximage Limited (IE) 2010-01-14 US disclosed
EP-2099742-A1 METHODS FOR PREPARING 2-METHOXYISOBUTYLISONITRILE AND TETRAKIS(2-METHOXYISOBUTYLISONITRILE)COPPER(I) TETRAFLUOROBORATE Draximage Limited (IE) 2009-09-16 EP disclosed
US-7563920-B2 Methods for preparing 2-methoxyisobutylisonitrile and tetrakis(2-methoxyisobutylisonitrile)copper(I) tetrafluoroborate Draximage Limited (IE) 2009-07-21 US disclosed
US-7563920-B2 Methods for preparing 2-methoxyisobutylisonitrile and tetrakis(2-methoxyisobutylisonitrile)copper(I) tetrafluoroborate Draximage Limited (IE) 2009-07-21 US disclosed
US-7563920-B2 Methods for preparing 2-methoxyisobutylisonitrile and tetrakis(2-methoxyisobutylisonitrile)copper(I) tetrafluoroborate Draximage Limited (IE) 2009-07-21 US disclosed
US-5652247-A VASOPRESSIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD (JP) 1997-07-29 US disclosed
US-5559230-A VASOPRESSIN ANTAGONISTS, QUINOLINES, BENZAZEPINES, VASODILATION, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-09-24 US disclosed
EP-0450097-B1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMA CO LTD (JP) 1996-04-24 EP disclosed
US-5498609-A Benzoazepinyl compounds as oxytocin and vasopressin antagonists OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1996-03-12 US disclosed
US-5436254-A Vaopressin antagonists OTSUKA PHARMACEUTICAL COMPANY, LTD. (JP) 1995-07-25 US disclosed
EP-0602209-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-22 EP disclosed
EP-0382185-B1 Carbostyril derivatives OTSUKA PHARMA CO LTD (JP) 1994-06-15 EP disclosed
WO-1994001113-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-01-20 WO disclosed
US-5225402-A Vasopressin antagonist, vasodilation, hypotensive, diuretics and anticoagulants OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-07-06 US disclosed
WO-1991005549-A1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-05-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100010250-A1 METHODS FOR PREPARING 2-METHOXYISOBUTYLISONITRILE AND TETRAKIS(2-METHOXYISOBUTYLISONITRILE)COPPER(I) TETRAFLUOROBORATE MEN1, CYP2F1, CYP4F11 ALDH1A1 2915/4885CHRM2 3470/4885CA12 1161/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.