SCHEMBL3170774

SCHEMBL3170774

CCOC(=O)CC(=O)c1ccc(OCc2ccccc2)c(OC)c1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.73
NPC1 O15118 2/20 0.73
RAB9A P51151 2/20 0.73
HPGD P15428 1/20 0.73
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
MAPT P10636 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
SMPD1 P17405 2/20 0.58
HDAC1 Q13547 1/20 0.58
HDAC8 Q9BY41 1/20 0.58
HDAC6 Q9UBN7 1/20 0.58
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
KDM4E B2RXH2 2/20 0.57
ALDH1A1 P00352 1/20 0.55
ABCB1 P08183 1/20 0.55
MRGPRX4 Q96LA9 1/20 0.53
APP P05067 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30951580 1.00 SMN1; SMN2 (0.73) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL3168608 0.95 SMN1; SMN2 (0.66) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL30100601 0.94 SMN1; SMN2 (0.63) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL21902756 0.94 SMN1; SMN2 (0.63) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL4872484 0.90 SMN1; SMN2 (0.76) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL6483625 0.88 SMN1; SMN2 (0.55) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL1034120 0.88 NPC1 (0.55) SMN1; SMN2NPC1RAB9AHPGDMAPT
SCHEMBL6246974 0.86 SMN1; SMN2 (0.78) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL3178525 0.86 HPGD (0.53) SMN1; SMN2NPC1RAB9AHPGDCYP1A2
SCHEMBL340393 0.85 SMN1; SMN2 (0.72) SMN1; SMN2NPC1RAB9AHPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645772-B2 4-(4-benzyloxy-3-chlorophenyl)-4-oxobutanoic acid; Methyl 4-(4-benzyloxy-2-methoxyphenyl)-4-oxobutanoate or derivatives for treatment of insulin resistance syndrome, diabetes, cachexia, hyperlipidemia, fatty liver disease, obesity, atherosclerosis or arteriosclerosis WELLSTAT THERAPEUTICS CORPORATION (US) 2010-01-12 US claimed
US-20060035970-A1 Compounds for the treatment of metabolic disorders WELLSTAT THERAPEUTICS CORPORATION 2006-02-16 US claimed
EP-1556085-A2 COMPOUNDS FOR THE TREATMENT OF METABOLIC DISORDERS Wellstat Therapeutics Corporation (US) 2005-07-27 EP claimed
WO-2004041165-A2 COMPOUNDS FOR THE TREATMENT OF METABOLIC DISORDERS WELLSTAT THERAPEUTICS CORPORATION (US) 2004-05-21 WO claimed
CN-118076605-A Substituted 1H-pyrazolo [4,3-c ] quinolines, methods of preparation and uses thereof 洛蒙治疗公司 2024-05-24 CN disclosed
US-7645772-B2 4-(4-benzyloxy-3-chlorophenyl)-4-oxobutanoic acid; Methyl 4-(4-benzyloxy-2-methoxyphenyl)-4-oxobutanoate or derivatives for treatment of insulin resistance syndrome, diabetes, cachexia, hyperlipidemia, fatty liver disease, obesity, atherosclerosis or arteriosclerosis WELLSTAT THERAPEUTICS CORPORATION (US) 2010-01-12 US disclosed
US-20060035970-A1 Compounds for the treatment of metabolic disorders WELLSTAT THERAPEUTICS CORPORATION 2006-02-16 US disclosed
EP-1556085-A2 COMPOUNDS FOR THE TREATMENT OF METABOLIC DISORDERS Wellstat Therapeutics Corporation (US) 2005-07-27 EP disclosed
WO-2004041165-A2 COMPOUNDS FOR THE TREATMENT OF METABOLIC DISORDERS WELLSTAT THERAPEUTICS CORPORATION (US) 2004-05-21 WO disclosed