SCHEMBL3171007

SCHEMBL3171007

CC(=O)NCCNc1cc(N2CCN(C(=O)c3cnccn3)CC2)nc(-c2ccccc2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM6B O15054 3/20 0.50
KDM2B Q8NHM5 3/20 0.50
CHRNA1 P02708 2/20 0.50
MAOB P27338 2/20 0.50
OPRM1 P35372 2/20 0.50
OPRK1 P41145 2/20 0.50
PDE4B Q07343 2/20 0.50
SCN5A Q14524 2/20 0.50
KDM4C Q9H3R0 2/20 0.50
KDM5B Q9UGL1 2/20 0.50
PHF8 Q9UPP1 2/20 0.50
NR1I2 O75469 1/20 0.50
AHR P35869 1/20 0.50
AVPR1A P37288 1/20 0.50
SLCO1B1 Q9Y6L6 1/20 0.50
GBA1 P04062 1/20 0.49
HDAC1 Q13547 3/20 0.47
HDAC6 Q9UBN7 3/20 0.47
SLC6A7 Q99884 1/20 0.46
CYP1A2 P05177 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3175655 0.92 GBA1 (0.47) KDM6BKDM2BCHRNA1MAOBOPRM1
SCHEMBL3170371 0.91 KDM6A (0.48) KDM6BKDM2BCHRNA1MAOBOPRM1
SCHEMBL3161894 0.89 ALDH1A1 (0.47) KDM6BKDM2BCHRNA1MAOBOPRM1
SCHEMBL3163116 0.88 KDM6B (0.50) KDM6BKDM2BCHRNA1MAOBOPRM1
SCHEMBL3164783 0.87 KDM6B (0.45) KDM6BKDM2BCHRNA1MAOBOPRM1
SCHEMBL3258026 0.87 PTK2 (0.46) KDM6BKDM2BCHRNA1MAOBOPRM1
SCHEMBL3155347 0.86 GBA1 (0.49) KDM6BKDM2BCHRNA1MAOBOPRM1
SCHEMBL3166309 0.86 GBA1 (0.48) KDM6BKDM2BCHRNA1MAOBOPRM1
SCHEMBL3171321 0.85 GBA1 (0.54) KDM6BKDM2BCHRNA1MAOBOPRM1
SCHEMBL3165783 0.85 USP2 (0.43) KDM6BKDM2BCHRNA1MAOBOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465631-B1 PYRIMIDINE A2B SELECTIVE ANTAGONIST COMPOUNDS, THEIR SYNTHESIS AND USE OSI PHARM INC (US) 2010-02-24 EP disclosed