SCHEMBL3172317

SCHEMBL3172317

CC(=O)NCCNc1nc(-c2ccccc2)nc(NCCNC(=O)c2cccc(C(F)(F)F)c2)c1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.53
ADORA1 P30542 1/20 0.53
ALDH1A1 P00352 5/20 0.53
POLB P06746 1/20 0.53
RXFP1 Q9HBX9 1/20 0.50
ADORA3 P0DMS8 1/20 0.49
TP53BP1 Q12888 1/20 0.48
CYP1A2 P05177 6/20 0.48
CYP3A4 P08684 6/20 0.48
CYP2D6 P10635 5/20 0.48
CLK4 Q9HAZ1 4/20 0.48
TSHR P16473 4/20 0.48
CYP2C19 P33261 2/20 0.48
USP2 O75604 2/20 0.47
MAPT P10636 3/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.46
ALOX15 P16050 1/20 0.46
RECQL P46063 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3172362 0.92 ALDH1A1 (0.50) ADORA2AADORA1ALDH1A1POLBRXFP1
SCHEMBL3258726 0.90 ADORA2A (0.57) ADORA2AADORA1ALDH1A1POLBRXFP1
SCHEMBL3162869 0.88 ALDH1A1 (0.55) ALDH1A1POLBRXFP1ADORA3TP53BP1
SCHEMBL3175889 0.87 ADORA2A (0.58) ADORA2AADORA1ALDH1A1POLBCYP1A2
SCHEMBL3165096 0.86 ADORA2A (0.65) ADORA2AADORA1ALDH1A1POLBCYP1A2
SCHEMBL3177178 0.85 ADORA2A (0.56) ADORA2AADORA1ALDH1A1TP53BP1CYP1A2
SCHEMBL3166454 0.83 ADORA2A (0.56) ADORA2AADORA1ALDH1A1POLBCYP1A2
SCHEMBL3162050 0.83 ADORA2A (0.72) ADORA2AADORA1ALDH1A1CYP1A2CYP3A4
SCHEMBL3165028 0.83 ADORA2A (0.58) ADORA2AADORA1ALDH1A1POLBCYP1A2
SCHEMBL3256770 0.82 CYP1A2 (0.67) ADORA2AADORA1ALDH1A1POLBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465631-B1 PYRIMIDINE A2B SELECTIVE ANTAGONIST COMPOUNDS, THEIR SYNTHESIS AND USE OSI PHARM INC (US) 2010-02-24 EP disclosed