SCHEMBL3175693

SCHEMBL3175693

CC(=O)NCCNc1cc(N2CCN(C(=O)c3ccc4cc(O)ccc4c3)CC2)nc(-c2ccccc2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.45
ALDH1A1 P00352 3/20 0.45
HTT P42858 2/20 0.45
USP2 O75604 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
ALOX15 P16050 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
POLB P06746 1/20 0.43
GBA1 P04062 2/20 0.43
KDM6B O15054 3/20 0.43
KDM2B Q8NHM5 3/20 0.43
CHRNA1 P02708 2/20 0.43
MAOB P27338 2/20 0.43
OPRM1 P35372 2/20 0.43
OPRK1 P41145 2/20 0.43
PDE4B Q07343 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3172676 0.92 GBA1 (0.43) LMNAALDH1A1HTTUSP2GAA
SCHEMBL3175804 0.91 GBA1 (0.51) LMNAALDH1A1MEN1KMT2APOLB
SCHEMBL3171321 0.89 GBA1 (0.54) LMNAALDH1A1MEN1KMT2APOLB
SCHEMBL3155347 0.89 GBA1 (0.49) LMNAALDH1A1GBA1KDM6BKDM2B
SCHEMBL3166309 0.88 GBA1 (0.48) LMNAALDH1A1HTTMAPTGBA1
SCHEMBL3163092 0.88 KDM6B (0.43) LMNAALDH1A1USP2MAPTPOLB
SCHEMBL3172356 0.88 GBA1 (0.45) LMNAALDH1A1MAPTALOX15HSD17B10
SCHEMBL3163851 0.88 GBA1 (0.48) LMNAALDH1A1POLBGBA1KDM6B
SCHEMBL3172414 0.88 GBA1 (0.50) LMNAALDH1A1MAPTMEN1KMT2A
SCHEMBL3175858 0.87 SLC6A7 (0.48) LMNAALDH1A1USP2MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465631-B1 PYRIMIDINE A2B SELECTIVE ANTAGONIST COMPOUNDS, THEIR SYNTHESIS AND USE OSI PHARM INC (US) 2010-02-24 EP disclosed