SCHEMBL3176404

SCHEMBL3176404

COc1cccc(-n2nc(C(C)(C)C)cc2NC(=O)OCC(Cl)(Cl)Cl)c1

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 12/20 0.64
MAPK13 O15264 5/20 0.64
MAPK12 P53778 5/20 0.64
MAPK11 Q15759 5/20 0.64
JAK2 O60674 1/20 0.52
MAPK9 P45984 3/20 0.48
DDR2 Q16832 3/20 0.48
GAA P10253 2/20 0.48
HPGD P15428 1/20 0.48
NTRK1 P04629 1/20 0.47
NTRK2 Q16620 1/20 0.47
CDK8 P49336 1/20 0.47
RECQL P46063 1/20 0.47
SRC P12931 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3187909 0.90 MAPK14 (0.61) MAPK14MAPK13MAPK12MAPK11JAK2
SCHEMBL26933627 0.90 MAPK14 (0.55) MAPK14MAPK13MAPK12MAPK11JAK2
SCHEMBL2452394 0.89 MAPK14 (0.62) MAPK14MAPK13MAPK12MAPK11JAK2
SCHEMBL3174914 0.88 MAPK14 (0.50) MAPK14MAPK13MAPK12MAPK11JAK2
SCHEMBL2361698 0.88 JAK2 (0.66) MAPK14MAPK13MAPK12MAPK11JAK2
SCHEMBL13532240 0.88 JAK2 (0.50) MAPK14MAPK13MAPK12MAPK11JAK2
SCHEMBL4420318 0.88 MAPK14 (0.60) MAPK14MAPK13MAPK12MAPK11JAK2
SCHEMBL15025600 0.88 MAPK14 (0.49) MAPK14MAPK13MAPK12MAPK11JAK2
SCHEMBL15007939 0.88 MAPK14 (0.49) MAPK14MAPK13MAPK12MAPK11JAK2
SCHEMBL15006941 0.88 MAPK14 (0.49) MAPK14MAPK13MAPK12MAPK11JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3999057-A1 POLYAROMATIC UREA DERIVATIVES AND THEIR USE IN THE TREATMENT OF MUSCLE DISEASES ANAGENESIS BIOTECHNOLOGIES SAS (FR) 2022-05-25 EP disclosed
US-20100016319-A1 ARYLMETHYLENE UREA DERIVATIVE AND USE THEREOF TORAY INDUSTRIES, INC. A CORPORATION OF JAPAN (JP) 2010-01-21 US disclosed
US-20100016319-A1 ARYLMETHYLENE UREA DERIVATIVE AND USE THEREOF TORAY INDUSTRIES, INC. A CORPORATION OF JAPAN (JP) 2010-01-21 US disclosed
US-20100016319-A1 ARYLMETHYLENE UREA DERIVATIVE AND USE THEREOF TORAY INDUSTRIES, INC. A CORPORATION OF JAPAN (JP) 2010-01-21 US disclosed
EP-1970375-A1 ARYLMETHYLENE UREA DERIVATIVE AND USE THEREOF TORAY INDUSTRIES, INC. (JP) 2008-09-17 EP disclosed
EP-1970375-A1 ARYLMETHYLENE UREA DERIVATIVE AND USE THEREOF TORAY INDUSTRIES, INC. (JP) 2008-09-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100016319-A1 ARYLMETHYLENE UREA DERIVATIVE AND USE THEREOF UROD, UTS2R, SLC14A1 MAPK14 500/4885MAPK13 593/4885MAPK12 1129/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.