SCHEMBL317924

SCHEMBL317924

C[C@@]12CCC[C@H]1[C@@H]1CCC3CCCC[C@]3(C)[C@@H]1CC2

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 1/20 0.64
CDK5R1 Q15078 1/20 0.64
NR1I3 Q14994 1/20 0.64
CYP19A1 P11511 3/20 0.56
GRIN1 Q05586 7/20 0.54
GRIN2B Q13224 7/20 0.54
MBOAT4 Q96T53 2/20 0.46
EPHA2 P29317 2/20 0.45
AKR1B10 O60218 1/20 0.45
AKR1B1 P15121 1/20 0.45
EFNA1 P20827 1/20 0.45
PSEN1 P49768 1/20 0.45
PSEN2 P49810 1/20 0.45
GPBAR1 Q8TDU6 1/20 0.45
APH1B Q8WW43 1/20 0.45
NCSTN Q92542 1/20 0.45
APH1A Q96BI3 1/20 0.45
PSENEN Q9NZ42 1/20 0.45
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4998837 1.00 CDK5 (0.64) CDK5CDK5R1NR1I3CYP19A1GRIN1
SCHEMBL157802 1.00 CDK5 (0.64) CDK5CDK5R1NR1I3CYP19A1GRIN1
SCHEMBL30331615 1.00 CDK5 (0.64) CDK5CDK5R1NR1I3CYP19A1GRIN1
SCHEMBL474980 1.00 CDK5 (0.64) CDK5CDK5R1NR1I3CYP19A1GRIN1
SCHEMBL157803 1.00 CDK5 (0.64) CDK5CDK5R1NR1I3CYP19A1GRIN1
SCHEMBL24451237 1.00 CDK5 (0.64) CDK5CDK5R1NR1I3CYP19A1GRIN1
SCHEMBL4998832 1.00 CDK5 (0.64) CDK5CDK5R1NR1I3CYP19A1GRIN1
SCHEMBL10343473 1.00 CDK5 (0.64) CDK5CDK5R1NR1I3CYP19A1GRIN1
SCHEMBL11241858 0.98 CDK5 (0.62) CDK5CDK5R1NR1I3CYP19A1GRIN1
Hydrochloric Acid SCHEMBL1591866 0.98 CDK5 (0.62) CDK5CDK5R1NR1I3CYP19A1GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 78 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1724554-A 1,4-pregnandiene 17 alpha, 21'-dihydroxy-3,20-diketone-17 alpha, 21-diacetate UNIV SICHUAN (CN) 2006-01-25 CN claimed
EP-1379542-A2 TREATMENT OF TUMOURS Hagström, Tomas (SE) 2004-01-14 EP claimed
WO-2002072003-A2 USE OF STEROID DERIVATIVES FOR THE TREATMENT OF A BENIGHN AND/OR MALIGNANT TUMOUR HAGSTROEM TOMAS (SE) 2002-09-19 WO claimed
CN-117281815-A Asymmetric synthesis and use of compounds in the treatment of disease 浙江嘉驰医药开发有限公司 2023-12-26 CN disclosed
CN-117281816-A Asymmetric synthesis and use of compounds in the treatment of disease 浙江嘉驰医药开发有限公司 2023-12-26 CN disclosed
EP-3681504-B1 METHODS OF DETECTION USING X-RAY FLUORESCENCE ICAGEN INC (US) 2023-08-23 EP disclosed
CN-111050771-B Asymmetric synthesis and use of compounds in the treatment of disease 浙江嘉驰医药开发有限公司 2023-08-01 CN disclosed
US-11573224-B2 Methods of detection using X-ray fluorescence ICAGEN, LLC (US) 2023-02-07 US disclosed
CN-109503691-A A kind of synthetic method of 5 α-androstane -3,17- diketone 华中药业股份有限公司 2019-03-22 CN disclosed
CN-107619424-A A kind of preparation method of 17 hydroxyl nitrile steroid derivative 天津金耀集团有限公司 2018-01-23 CN disclosed
US-9868757-B2 5-β, 14-β-androstane derivatives useful for the treatment of proteinuria, glomerulosclerosis and renal failure SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 2018-01-16 US disclosed
CN-1100101-A 14alpha-hydroxy-4-androstene-3,6,17-trione hydrate crystal and process for producing same NIPPON KAYAKU KK (JP) 1995-03-15 CN disclosed
CN-1026236-C Steroid 5-alpha-reductase inhibitors SMITHKLINE BECKMAN CORP (US) 1994-10-19 CN disclosed
EP-0583606-A2 New hydrazono-5-beta-androstane derivatives active on the cardiovascular system, processes for their preparation and pharmaceutical compositions containing same Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. (IT) 1994-02-23 EP disclosed
CN-1079747-A The preparation of pharmaceutical compositions method that contains steroid 5-alpha-reductase inhibitors SMITHKLINE BECKAMAN CORP (US) 1993-12-22 CN disclosed
CN-1071418-A Benzo [ f ] quinolinones LILLY CO ELI (US) 1993-04-28 CN disclosed
EP-0253415-B1 PROCESS FOR THE PREPARATION OF 9(11)-DEHYDROANDROSTANES GIST-BROCADES N.V. (NL) 1990-03-14 EP disclosed
CN-1030765-A STEROID 5-ALPHA-REDUCTASE INHIBITORS SMITHKLINE BECKMAN CORP (US) 1989-02-01 CN disclosed
EP-0253415-A1 Process for the preparation of 9(11)-dehydroandrostanes GIST-BROCADES N.V. (NL) 1988-01-20 EP disclosed
US-4075233-A SKIN DISORDERS GIST-BROCADES N.V. (NL) 1978-02-21 US disclosed