SCHEMBL3196293

SCHEMBL3196293

CC(O)c1cc(=O)oc2cc3c(cc12)CCCN3

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 3/20 0.67
AR P10275 7/20 0.59
KDM4E B2RXH2 8/20 0.41
ALDH1A1 P00352 6/20 0.41
GLA P06280 3/20 0.41
GAA P10253 3/20 0.41
HPGD P15428 3/20 0.41
CASP1 P29466 3/20 0.41
CASP7 P55210 3/20 0.41
HSD17B10 Q99714 3/20 0.41
KMT2A Q03164 3/20 0.39
PGR P06401 4/20 0.37
NR3C2 P08235 1/20 0.37
HCAR2 Q8TDS4 1/20 0.36
LMNA P02545 3/20 0.36
MAPT P10636 3/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29580428 0.80 ATM (1.00) ATMARKDM4EALDH1A1GLA
SCHEMBL17717500 0.80 ATM (1.00) ATMARKDM4EALDH1A1GLA
SCHEMBL3196150 0.79 ATM (0.68) ATMARKDM4EALDH1A1GLA
SCHEMBL29474210 0.74 AR (1.00) ATMARCASP1CASP7KMT2A
SCHEMBL3262044 0.74 KDM4E (0.47) ATMARKDM4EALDH1A1GLA
SCHEMBL22100626 0.73 ATM (0.61) ATMARKDM4EALDH1A1GLA
SCHEMBL11028692 0.72 ATM (0.84) ATMARKDM4EALDH1A1GLA
SCHEMBL5233514 0.71 AR (0.93) ATMARCASP1CASP7KMT2A
SCHEMBL17717371 0.70 ATM (0.64) ATMARKDM4EALDH1A1GLA
SCHEMBL11552058 0.69 ATM (0.58) ATMARKDM4EALDH1A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100048604-A1 Ligands for Aldoketoreductases TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2010-02-25 US disclosed
US-20100048604-A1 Ligands for Aldoketoreductases TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2010-02-25 US disclosed
US-20100048604-A1 Ligands for Aldoketoreductases TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2010-02-25 US disclosed
WO-2006023821-A2 LIGANDS FOR ALDOKETOREDUCTASES THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2006-03-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048604-A1 Ligands for Aldoketoreductases AKR1C2, AKR1C1, AKR1B1 ATM 3509/4885AR 182/4885KDM4E 2592/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.