SCHEMBL320618

SCHEMBL320618

[CH]c1ccc(-c2noc(-c3ccc(-c4ccccc4C)c(COC)c3)n2)cc1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 17/20 0.67
S1PR3 Q99500 2/20 0.67
NR1H4 Q96RI1 1/20 0.48
NPC1 O15118 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MAPT P10636 1/20 0.47
PKM P14618 1/20 0.47
NFKB1 P19838 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TP53 P04637 1/20 0.46
GAA P10253 1/20 0.46
MAPK1 P28482 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL320617 1.00 S1PR1 (0.67) S1PR1S1PR3NR1H4NPC1SMN1; SMN2
SCHEMBL320619 0.91 S1PR1 (0.69) S1PR1S1PR3NR1H4NPC1SMN1; SMN2
SCHEMBL320407 0.87 S1PR1 (0.70) S1PR1S1PR3NR1H4NPC1SMN1; SMN2
SCHEMBL14916846 0.86 S1PR1 (0.67) S1PR1S1PR3NR1H4NPC1SMN1; SMN2
SCHEMBL2806793 0.85 S1PR1 (0.71) S1PR1S1PR3NR1H4NPC1SMN1; SMN2
SCHEMBL410568 0.85 S1PR1 (0.68) S1PR1S1PR3NR1H4NPC1SMN1; SMN2
SCHEMBL15905722 0.85 S1PR1 (0.64) S1PR1S1PR3NR1H4NPC1SMN1; SMN2
SCHEMBL13187540 0.85 S1PR1 (0.67) S1PR1S1PR3NR1H4NPC1SMN1; SMN2
SCHEMBL409297 0.85 S1PR1 (0.66) S1PR1S1PR3NR1H4NPC1SMN1; SMN2
SCHEMBL407139 0.84 S1PR1 (0.66) S1PR1S1PR3NR1H4NPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590956-A1 5-(BIPHENYL-4-YL)-3-PHENYL-1,2,4-OXADIAZOLYL DERIVATIVES AS LIGANDS ON THE SPHINGOSINE 1-PHOSPHATE (S1P) RECEPTORS Merck Serono S.A. (CH) 2013-05-15 EP disclosed
WO-2012004287-A1 5-(BIPHENYL-4-YL)-3-PHENYL-1,2,4-OXADIAZOLYL DERIVATIVES AS LIGANDS ON THE SPHINGOSINE 1-PHOSPHATE (S1P) RECEPTORS MERCK SERONO S.A. (CH) 2012-01-12 WO disclosed