SCHEMBL320619

SCHEMBL320619

COCc1cc(-c2nc(-c3ccc(C)cc3)no2)ccc1-c1ccccc1C

nearest known ligand 0.69

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 16/20 0.69
S1PR3 Q99500 2/20 0.69
NPC1 O15118 2/20 0.52
NFKB1 P19838 2/20 0.52
RAB9A P51151 2/20 0.52
NFKB2 Q00653 2/20 0.52
RELA Q04206 2/20 0.52
MAPK1 P28482 2/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
TP53 P04637 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
NR1H4 Q96RI1 1/20 0.50
TSHR P16473 1/20 0.50
TDP1 Q9NUW8 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL320617 0.91 S1PR1 (0.67) S1PR1S1PR3NPC1NFKB1RAB9A
SCHEMBL320618 0.91 S1PR1 (0.67) S1PR1S1PR3NPC1NFKB1RAB9A
SCHEMBL320407 0.89 S1PR1 (0.70) S1PR1S1PR3NPC1NFKB1NFKB2
SCHEMBL14916846 0.88 S1PR1 (0.67) S1PR1S1PR3NPC1NFKB1RAB9A
SCHEMBL9968839 0.87 S1PR1 (0.65) S1PR1S1PR3NPC1NFKB1RAB9A
SCHEMBL2806793 0.87 S1PR1 (0.71) S1PR1S1PR3NPC1NFKB1RAB9A
SCHEMBL410568 0.87 S1PR1 (0.68) S1PR1S1PR3NPC1NFKB1RAB9A
SCHEMBL15905722 0.87 S1PR1 (0.64) S1PR1S1PR3NPC1NFKB1RAB9A
SCHEMBL13187540 0.87 S1PR1 (0.67) S1PR1S1PR3NPC1NFKB1RAB9A
SCHEMBL409297 0.87 S1PR1 (0.66) S1PR1S1PR3NPC1NFKB1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590956-A1 5-(BIPHENYL-4-YL)-3-PHENYL-1,2,4-OXADIAZOLYL DERIVATIVES AS LIGANDS ON THE SPHINGOSINE 1-PHOSPHATE (S1P) RECEPTORS Merck Serono S.A. (CH) 2013-05-15 EP disclosed
WO-2012004287-A1 5-(BIPHENYL-4-YL)-3-PHENYL-1,2,4-OXADIAZOLYL DERIVATIVES AS LIGANDS ON THE SPHINGOSINE 1-PHOSPHATE (S1P) RECEPTORS MERCK SERONO S.A. (CH) 2012-01-12 WO disclosed