SCHEMBL3208247

SCHEMBL3208247

NC1=c2ncn([C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)c2=NCN1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.51
ALDH1A1 P00352 2/20 0.51
HTT P42858 2/20 0.51
BLM P54132 2/20 0.51
LMNA P02545 2/20 0.51
GMNN O75496 1/20 0.51
NFKB1 P19838 1/20 0.51
DNMT1 P26358 1/20 0.51
THPO P40225 1/20 0.51
MTOR P42345 1/20 0.51
RAB9A P51151 1/20 0.51
HBB P68871 1/20 0.51
PMP22 Q01453 1/20 0.51
KDM4E B2RXH2 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
MAPT P10636 1/20 0.50
ADORA2A P29274 3/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
ADORA3 P0DMS8 2/20 0.49
ADORA2B P29275 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6704178 0.88 TP53 (0.51) TP53ALDH1A1HTTBLMLMNA
SCHEMBL136036 0.88 TP53 (0.51) TP53ALDH1A1HTTBLMLMNA
SCHEMBL40771 0.87 TP53 (0.50) TP53ALDH1A1HTTBLMLMNA
SCHEMBL5317002 0.87 TP53 (0.50) TP53ALDH1A1HTTBLMLMNA
SCHEMBL7145382 0.83 TP53 (0.50) TP53ALDH1A1HTTBLMLMNA
SCHEMBL16333894 0.82 TP53 (0.45) TP53ALDH1A1HTTBLMLMNA
SCHEMBL4406383 0.81 TP53 (0.47) TP53ALDH1A1HTTBLMLMNA
SCHEMBL4271353 0.80 TP53 (0.46) TP53ALDH1A1HTTBLMLMNA
SCHEMBL2809573 0.80 TP53 (0.46) TP53ALDH1A1HTTBLMLMNA
SCHEMBL5507731 0.80 TP53 (0.43) TP53ALDH1A1HTTBLMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-57206396-A None JP disclosed
US-7666646-B2 Crystal structure of human Pim-1 kinase protein complexes and binding pockets thereof, and uses thereof in drug design VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-02-23 US disclosed
US-20070031956-A1 Crystal structure of human PIM-1 kinase protein complexes and binding pockets thereof, and uses thereof in drug design VERTEX PHARMACEUTICALS INCORPORATED 2007-02-08 US disclosed
JP-S57206396-A PREPARATION OF CYCLIC-3',5'-ADENYLIC ACID BY FERMENTATION METHOD KIKKOMAN CORP 1982-12-17 JP disclosed