SCHEMBL3225657

SCHEMBL3225657

N#CC(=O)Cc1ccncc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 10/20 0.44
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
KDM4E B2RXH2 1/20 0.41
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL955096 0.78 CES1 (0.56) ALDH1A1GAAHDAC6
SCHEMBL4594374 0.77 NAPRT (0.62) CYP19A1ALDH1A1GAAKDM4E
SCHEMBL13799024 0.77 CA2 (0.56) ALDH1A1KDM4ERAB9ANPC1CA2
SCHEMBL10520154 0.76 CYP19A1 (0.42) CYP19A1ALDH1A1GAAMAPTRAB9A
SCHEMBL10445460 0.75 NPC1 (0.47) ALDH1A1MAPTRAB9ANPC1SMN1; SMN2
SCHEMBL10172435 0.75 GAA (0.48) ALDH1A1GAAKDM4ERAB9ASMN1; SMN2
SCHEMBL11470932 0.75 CTBP2 (0.47) ALDH1A1GAARAB9ANPC1SMN1; SMN2
SCHEMBL10750108 0.75 CYP19A1 (0.52) CYP19A1ALDH1A1GAAMAPTKDM4E
SCHEMBL8040203 0.73 CYP19A1 (0.50) CYP19A1ALDH1A1GAAMAPTKDM4E
SCHEMBL48554 0.73 AKR1B1 (0.61) CYP19A1ALDH1A1GAAMAPTCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010009290-A1 ALPHA7 NICOTINIC ACETYLCHOLINE RECEPTOR INHIBITORS WYETH (US) 2010-01-21 WO disclosed