SCHEMBL3225890

SCHEMBL3225890

C=C1C[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1C(C)=O

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 9/20 0.66
SHBG P04278 8/20 0.66
SMN1; SMN2 Q16637 7/20 0.66
SERPINA6 P08185 7/20 0.66
CYP3A4 P08684 6/20 0.66
MAPK1 P28482 6/20 0.66
ALDH1A1 P00352 6/20 0.66
TSHR P16473 5/20 0.66
MAPT P10636 5/20 0.66
NR3C1 P04150 4/20 0.66
PGR P06401 3/20 0.66
AR P10275 3/20 0.66
GPBAR1 Q8TDU6 3/20 0.66
SIGMAR1 Q99720 3/20 0.66
PMP22 Q01453 3/20 0.66
NPSR1 Q6W5P4 3/20 0.66
CYP2C9 P11712 2/20 0.66
HIF1A Q16665 2/20 0.66
CYP2C19 P33261 2/20 0.66
MEN1 O00255 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3671789 0.89 LMNA (0.69) LMNASHBGSMN1; SMN2SERPINA6CYP3A4
SCHEMBL7242829 0.81 LMNA (0.58) LMNASHBGSMN1; SMN2SERPINA6CYP3A4
SCHEMBL6840982 0.81 CYP3A4 (0.55) LMNASHBGSMN1; SMN2SERPINA6CYP3A4
SCHEMBL6840979 0.81 CYP3A4 (0.55) LMNASHBGSMN1; SMN2SERPINA6CYP3A4
Progesterone SCHEMBL11659276 0.80 CYP3A4 (0.95) LMNASHBGSMN1; SMN2SERPINA6CYP3A4
Progesterone SCHEMBL23568915 0.80 CYP3A4 (1.00) LMNASHBGSMN1; SMN2SERPINA6CYP3A4
Progesterone SCHEMBL15224316 0.80 CYP3A4 (1.00) LMNASHBGSMN1; SMN2SERPINA6CYP3A4
Progesterone SCHEMBL8430168 0.80 CYP3A4 (1.00) LMNASHBGSMN1; SMN2SERPINA6CYP3A4
Progesterone SCHEMBL20409003 0.80 CYP3A4 (1.00) LMNASHBGSMN1; SMN2SERPINA6CYP3A4
Progesterone SCHEMBL13259536 0.80 CYP3A4 (1.00) LMNASHBGSMN1; SMN2SERPINA6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8586080-B1 Inhibiting crystallization of steroidal hormones in transdermal delivery systems NOVEN PHARMACEUTICALS, INC. (US) 2013-11-19 US disclosed
US-20100047345-A1 HYDROPHOBIC ABUSE DETERRENT DELIVERY SYSTEM FOR HYDROMORPHONE CROWLEY MICHAEL M 2010-02-25 US disclosed
EP-2068840-A2 HYDROPHOBIC ABUSE DETERRENT DELIVERY SYSTEM LAB International SRL (US) 2009-06-17 EP disclosed
EP-2049087-A2 HYDROPHILIC ABUSE DETERRENT DELIVERY SYSTEM LAB International SRL (US) 2009-04-22 EP disclosed
US-20080075770-A1 HYDROPHILIC ABUSE DETERRENT DELIVERY SYSTEM AKELA PHARMA SRL (BB) 2008-03-27 US disclosed
US-20080075768-A1 HYDROPHOBIC OPIOID ABUSE DETERRENT DELIVERY SYSTEM USING OPIOID ANTAGONISTS AKELA PHARMA SRL (BB) 2008-03-27 US disclosed
US-20080069871-A1 HYDROPHOBIC ABUSE DETERRENT DELIVERY SYSTEM AKELA PHARMA SRL (BB) 2008-03-20 US disclosed
US-20080063698-A1 Crystallization inhibition of drugs in transdermal drug delivery systems and methods of use NOVEN PHARMACEUTICALS, INC. 2008-03-13 US disclosed
WO-2008011595-A9 HYDROPHOBIC ABUSE DETERRENT DELIVERY SYSTEM LAB INTERNAT SRL (US) 2008-03-06 WO disclosed
WO-2008011596-A2 HYDROPHILIC ABUSE DETERRENT DELIVERY SYSTEM LAB INTERNATIONAL SRL (US) 2008-01-24 WO disclosed
US-20040142023-A1 Crystallization inhibition of drugs in transdermal drug delivery systems and methods of use NOVEN PHARMACEUTICALS, INC. 2004-07-22 US disclosed
WO-2004050066-A1 MICROSPHERES AND RELATED PROCESSES AND PHARMACEUTICAL COMPOSITIONS THE UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 2004-06-17 WO disclosed
US-6638528-B1 Pressure-sensitive adhesive matrix comprising blend of polyacrylate, polysiloxane, polyisobutylene, polyisoprene, polyamide or polystyrene; and insoluble, non-adhesive ethyl cellulose; polyvinylpyrrolidone crystallization inhibitor NOVEN PHARMACEUTICALS, INC. 2003-10-28 US disclosed
US-20030152616-A1 Crystallization inhibition of drugs in transdermal drug delivery systems and methods of use NOVEN PHARMACEUTICALS, INC. 2003-08-14 US disclosed
US-6465004-B1 ESTERIFIED OR ACYLATED CELLULOSE TO STABILIZE THE CONCENTRATION OF THE ACTIVE AGENT IN THE COMPOSITION AND TO INHIBIT CRYSTAL FORMATION; PRESSURE-SENSITIVE ADHESIVE CARRIER; CELLULOSE ACETATE BUTYRATE NOVEN PHARMACEUTICALS, INC. 2002-10-15 US disclosed
US-20020106402-A1 Crystallization inhibition of drugs in transdermal drug delivery systems and methods of use NOVEN PHARMACEUTICALS, INC. 2002-08-08 US disclosed
WO-2002045701-A2 CRYSTALLIZATION INHIBITION OF DRUGS IN TRANSDERMAL DRUG DELIVERY SYSTEMS NOVEN PHARMACEUTICALS, INC. (US) 2002-06-13 WO disclosed
US-20020004065-A1 Compositions and methods to effect the release profile in the transdermal administration of active agents KANIOS DAVID (US) 2002-01-10 US disclosed
WO-2001052823-A2 COMPOSITIONS TO EFFECT THE RELEASE PROFILE IN THE TRANSDERMAL ADMINISTRATION OF DRUGS NOVEN PHARMACEUTICALS, INC. (US) 2001-07-26 WO disclosed
WO-2000074661-A2 SOLUBILITY ENHANCEMENT OF DRUGS IN TRANSDERMAL DRUG DELIVERY SYSTEMS AND METHODS OF USE NOVEN PHARMACEUTICALS, INC. (US) 2000-12-14 WO disclosed