SCHEMBL3228463

SCHEMBL3228463

O=C(O)c1cc(-c2ccc(O)cc2)nc2c(F)cccc12

nearest known ligand 0.69

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.69
POLB P06746 1/20 0.64
PDE10A Q9Y233 2/20 0.54
EPRS1 P07814 2/20 0.54
DHODH Q02127 4/20 0.52
KDM4E B2RXH2 2/20 0.51
LMNA P02545 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
AKR1C3 P42330 1/20 0.51
AKR1C2 P52895 1/20 0.51
AKR1C1 Q04828 1/20 0.51
HTT P42858 1/20 0.50
PPARA Q07869 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22471898 0.90 AURKA (0.78) AURKAPOLBPDE10AEPRS1DHODH
SCHEMBL24270274 0.89 AURKA (0.69) AURKAPOLBPDE10AEPRS1DHODH
SCHEMBL3234823 0.86 AURKA (0.65) AURKAPOLBPDE10AEPRS1DHODH
SCHEMBL23771105 0.85 AURKA (0.63) AURKAPOLBPDE10AEPRS1DHODH
SCHEMBL29617660 0.85 AURKA (0.63) AURKAPDE10AEPRS1DHODHKDM4E
SCHEMBL23590310 0.85 AURKA (0.63) AURKAPDE10AEPRS1DHODHKDM4E
SCHEMBL24270273 0.84 AURKA (0.62) AURKAPDE10AEPRS1DHODHKDM4E
SCHEMBL25735926 0.82 AURKA (0.73) AURKAPDE10AEPRS1DHODHKDM4E
SCHEMBL24686630 0.82 AURKA (1.00) AURKAPOLBPDE10AEPRS1DHODH
SCHEMBL23590312 0.81 RAB9A (0.68) AURKAPOLBPDE10AEPRS1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010020672-A1 NOVEL PHENYL-QUINOLINE-CARBOXYLIC ACID PYRIDINE DERIVATIVES USEFUL AS MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS NEUROSEARCH A/S (DK) 2010-02-25 WO claimed
WO-2010020672-A1 NOVEL PHENYL-QUINOLINE-CARBOXYLIC ACID PYRIDINE DERIVATIVES USEFUL AS MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS NEUROSEARCH A/S (DK) 2010-02-25 WO disclosed