SCHEMBL3228656

SCHEMBL3228656

O=C(O)Oc1cn(Cc2cc(F)ccc2F)c2c(F)cccc2c1=O

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.47
P2RX7 Q99572 1/20 0.39
MAPT P10636 3/20 0.37
GAA P10253 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
TP53 P04637 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
ROCK2 O75116 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HPGD P15428 1/20 0.36
RORC P51449 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CNR2 P34972 1/20 0.36
MMP1 P03956 1/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
MMP12 P39900 1/20 0.35
RIPK1 Q13546 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3233811 0.91 CHRM1 (0.47) CHRM1P2RX7MAPTGAAPTGDR2
SCHEMBL3234252 0.88 CHRM1 (0.44) CHRM1P2RX7MAPTPTGDR2TP53
SCHEMBL3234223 0.86 CHRM1 (0.47) CHRM1P2RX7MAPTPTGDR2TP53
SCHEMBL3228651 0.85 CHRM1 (0.64) CHRM1MAPTTP53RXFP1
SCHEMBL3234555 0.85 CHRM1 (0.49) CHRM1P2RX7MAPTPTGDR2TP53
SCHEMBL3230518 0.84 CHRM1 (0.48) CHRM1MAPTGAAPTGDR2TP53
SCHEMBL3234268 0.84 CHRM1 (0.54) CHRM1P2RX7MAPTGAATP53
SCHEMBL3239684 0.84 CHRM1 (0.52) CHRM1P2RX7MAPTPTGDR2ROCK2
SCHEMBL3234589 0.83 CHRM1 (0.55) CHRM1P2RX7MAPTTP53SMN1; SMN2
SCHEMBL3234399 0.83 CHRM1 (0.63) CHRM1MAPTTP53CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-B1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK SHARP & DOHME (US) 2010-07-28 EP claimed