SCHEMBL3229200

SCHEMBL3229200

CC1(c2ccc(Cl)c(C(F)(F)F)c2)CC(CO[Si](c2ccccc2)(c2ccccc2)C(C)(C)C)CC=C1C(=O)O

nearest known ligand 0.73

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 19/20 0.73
OPRM1 P35372 1/20 0.37
OPRL1 P41146 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1779370 0.85 CCR2 (0.52) CCR2OPRM1OPRL1
SCHEMBL3233950 0.85 CCR2 (0.82) CCR2
SCHEMBL1780255 0.84 CCR2 (0.52) CCR2OPRM1OPRL1
SCHEMBL1780797 0.82 CCR2 (0.48) CCR2OPRM1OPRL1
SCHEMBL1780135 0.82 CCR2 (1.00) CCR2
SCHEMBL1781426 0.78 CCR2 (0.77) CCR2
SCHEMBL1781364 0.77 CCR2 (1.00) CCR2
SCHEMBL14237076 0.77 CCR2 (1.00) CCR2
SCHEMBL1779544 0.77 CCR2 (1.00) CCR2
SCHEMBL1780401 0.77 CCR2 (0.43) CCR2OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8507559-B2 Cyclohexenyl modulators of chemokine receptor activity BRISTOL-MYERS SQUIBB COMPANY (US) 2013-08-13 US disclosed
EP-2318352-B1 CYCLOHEXENYL COMPOUNDS AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2012-12-19 EP disclosed
WO-2010009068-A2 CYCLOHEXENYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2010-01-21 WO disclosed