SCHEMBL3233759

SCHEMBL3233759

CCN(c1ccccc1)c1cc(-c2ccccc2)nc(Nc2ccc(C3(C(=O)OC)CCC3)cc2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.38
MAPT P10636 2/20 0.37
AURKA O14965 1/20 0.36
PRCP P42785 2/20 0.36
SIGMAR1 Q99720 2/20 0.36
ALDH1A1 P00352 5/20 0.36
POLB P06746 1/20 0.36
ADORA1 P30542 4/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
IDO1 P14902 1/20 0.35
CHRM2 P08172 3/20 0.34
CHRM1 P11229 2/20 0.34
KDM4E B2RXH2 2/20 0.34
SLC22A1 O15245 1/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3227453 0.92 AURKA (0.38) MAPTAURKAALDH1A1ADORA1ADORA3
SCHEMBL3236000 0.90 AURKA (0.40) AKT1MAPTAURKAPRCPSIGMAR1
SCHEMBL3225921 0.85 ADORA1 (0.36) MAPTAURKAALDH1A1ADORA1ADORA3
SCHEMBL3232625 0.85 AKT1 (0.40) AKT1MAPTALDH1A1ADORA1ADORA3
SCHEMBL3221032 0.82 AURKA (0.41) MAPTAURKAALDH1A1ADORA1ADORA3
SCHEMBL3234072 0.81 AKT1 (0.46) AKT1MAPTADORA1ADORA3ADORA2A
SCHEMBL3227596 0.81 AKT1 (0.42) AKT1MAPTPOLBADORA1ADORA3
SCHEMBL13456904 0.79 VCP (0.48)
SCHEMBL3264602 0.78 AKT1 (0.40) AKT1MAPTADORA1ADORA3ADORA2A
SCHEMBL3228961 0.78 MAPT (0.47) AKT1MAPTPOLBLMNATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028179-A1 HETEROCYCLIC COMPOUNDS AS GATA MODULATORS DR. REDDY'S LABORATORIES LTD. (IN) 2010-03-11 WO disclosed