SCHEMBL3234085

SCHEMBL3234085

Nc1ccccc1NC(=O)OCC1c2ccccc2-c2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.58
EPHX2 P34913 1/20 0.57
FABP5 Q01469 3/20 0.47
FABP7 O15540 2/20 0.47
CHRM3 P20309 2/20 0.43
CHRM2 P08172 1/20 0.43
CHRM1 P11229 1/20 0.43
HDAC3 O15379 3/20 0.43
HDAC1 Q13547 3/20 0.43
HDAC2 Q92769 3/20 0.43
NCOR2 Q9Y618 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC9 Q9UKV0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17413389 0.84 EPHX2 (0.53) KMT2AEPHX2FABP5FABP7HDAC3
SCHEMBL31423769 0.84 EPHX2 (0.53) KMT2AEPHX2FABP5FABP7HDAC3
SCHEMBL29547309 0.84 EPHX2 (0.53) KMT2AEPHX2FABP5FABP7HDAC3
SCHEMBL14701886 0.84 EPHX2 (0.53) KMT2AEPHX2FABP5FABP7HDAC3
SCHEMBL29067330 0.83 EPHX2 (0.57) KMT2AEPHX2FABP5FABP7CHRM3
SCHEMBL20266541 0.83 KMT2A (0.52) KMT2AEPHX2FABP5FABP7HDAC3
SCHEMBL29019441 0.83 EPHX2 (0.49) KMT2AEPHX2FABP5FABP7CHRM3
SCHEMBL119223 0.82 EPHX2 (0.60) KMT2AEPHX2FABP5FABP7CHRM3
SCHEMBL29401765 0.82 EPHX2 (0.60) KMT2AEPHX2FABP5FABP7CHRM3
SCHEMBL29913938 0.82 EPHX2 (0.60) KMT2AEPHX2FABP5FABP7CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed