SCHEMBL3234136

SCHEMBL3234136

Cc1ncc2cccc(O)c2n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 2/20 0.55
KDM4E B2RXH2 10/20 0.55
MMP2 P08253 1/20 0.48
CHRM1 P11229 1/20 0.48
TSHR P16473 1/20 0.48
COMT P21964 1/20 0.48
ADRA1A P35348 1/20 0.48
METAP1 P53582 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
KMT2A Q03164 3/20 0.46
MEN1 O00255 1/20 0.46
PLAU P00749 1/20 0.46
NCF1 P14598 1/20 0.46
ALOX12 P18054 2/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8404376 0.79 CYP2A6 (0.39) KDM4EADRA1AALDH1A1CYP1A2
Lithium Ion SCHEMBL28782689 0.78 METAP2 (0.47) METAP2KDM4EMMP2CHRM1TSHR
SCHEMBL18630254 0.76 CYP1A2 (0.36) KDM4EKMT2AMEN1ALDH1A1CYP1A2
SCHEMBL3530216 0.76 NPC1 (0.38) KDM4EKMT2AMEN1ALDH1A1CYP1A2
SCHEMBL30881848 0.76 BACE1 (0.46) KDM4EALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL15691393 0.76 CYP1A2 (0.41) KDM4EKMT2ACYP1A2CYP2C9HPGD
SCHEMBL1632414 0.76 METAP2 (0.48) METAP2KDM4EMMP2CHRM1TSHR
SCHEMBL1634276 0.76 METAP2 (0.48) METAP2KDM4EMMP2CHRM1TSHR
SCHEMBL1041168 0.76 PLAU (0.55) METAP2KDM4EMMP2CHRM1TSHR
SCHEMBL28859362 0.76 METAP2 (0.48) METAP2KDM4EMMP2CHRM1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250381221-A1 Compositions and Methods for Treating Cancer IN8BIO INC (US) 2025-12-18 US disclosed
US-20240245643-A1 DNA Damage Repair Inhibitors for Treatment of Cancer THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL (GB) 2024-07-25 US disclosed
US-20220339179-A1 TREATMENT OF HR DEFICIENT CANCER THE FRANCIS CRICK INSTITUTE LIMITED (GB) 2022-10-27 US disclosed
EP-4028009-A1 TREATMENT OF HR DEFICIENT CANCER The Francis Crick Institute Limited (GB) 2022-07-20 EP disclosed
US-20220062286-A1 USE OF RNAI INHIBITING PARP ACTIVITY FOR THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF CANCER THE UNIVERSITY OF SHEFFIELD (GB) 2022-03-03 US disclosed
WO-2016164771-A1 METHODS OF CANCER DETECTION USING PARPi-FL MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2016-10-13 WO disclosed
CN-102762726-A Chimeric endonucleases and uses thereof BASF PLANT SCIENCE CO GMBH 2012-10-31 CN disclosed
CN-102725412-A Optimized endonucleases and uses thereof BASF PLANT SCIENCE CO GMBH 2012-10-10 CN disclosed
CN-102686726-A Chimeric endonucleases and uses thereof BASF PLANT SCIENCE CO GMBH 2012-09-19 CN disclosed
US-7998978-B2 Substituted 2-amino-fused heterocyclic compounds PFIZER INC. (US) 2011-08-16 US disclosed
US-6100284-A ANTIALLERGENS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-08 US disclosed
US-6008229-A TREATING ALLERGY, INFLAMMATION, AUTOIMMUNE DISEASE, SHOCK, PAIN FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-12-28 US disclosed
WO-1999064039-A1 BRADYKININ ANTAGONISTS ADVANCED MEDICINE, INC. (US) 1999-12-16 WO disclosed
US-5922711-A ANTIALLERGENS, ANTIINFLAMMATORY AGENTS, AUTOIMMUNE DISEASES, SHOCK OR ANALGESICS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-07-13 US disclosed
EP-0861243-A1 HETEROCYCLIC COMPOUNDS AS BRADYKININ ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-09-02 EP disclosed
US-5708173-A PREPARATION OF SUBSTITUTED QUINOLINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-01-13 US disclosed
WO-1997011069-A1 HETEROCYCLIC COMPOUNDS AS BRADYKININ ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-03-27 WO disclosed
US-5563162-A CAN BE ADMINISTERD FOR THE TREATMENT OF ALLERGY, INFLAMMATION, AUTOIMMUNE DISEASES, SHOCK OR PAIN IN ANIMALS AND HUMANS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-10-08 US disclosed
CN-1097417-A New heterogeneous ring compound FUJISAWA PHARMACEUTICAL CO (JP) 1995-01-18 CN disclosed
EP-0622361-A1 Heterocyclic compounds as bradykinin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-11-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240245643-A1 DNA Damage Repair Inhibitors for Treatment of Cancer PARP2, MRE11, PARP1 METAP2 2962/4885KDM4E 2660/4885MMP2 2612/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.