SCHEMBL3235002

SCHEMBL3235002

CC1COCCN1c1nc(-c2ccc3[nH]c(=O)ccc3c2)nc2c1CCN(C(=O)O)C2

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATR Q13535 6/20 0.54
MTOR P42345 14/20 0.51
KCNH2 Q12809 1/20 0.50
PIK3CA P42336 1/20 0.50
RPTOR Q8N122 4/20 0.48
MLST8 Q9BVC4 4/20 0.48
CYP3A4 P08684 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2097802 0.90 MTOR (0.59) ATRMTORKCNH2PIK3CARPTOR
SCHEMBL1830344 0.90 MTOR (0.59) ATRMTORKCNH2PIK3CARPTOR
SCHEMBL15189922 0.89 ATR (0.64) ATRMTORKCNH2PIK3CARPTOR
SCHEMBL1841030 0.87 MTOR (0.59) ATRMTORKCNH2PIK3CARPTOR
SCHEMBL1841028 0.87 MTOR (0.59) ATRMTORKCNH2PIK3CARPTOR
SCHEMBL3228564 0.82 ATR (0.53) ATRMTORKCNH2PIK3CARPTOR
SCHEMBL1841378 0.79 MTOR (0.60) ATRMTORKCNH2PIK3CARPTOR
SCHEMBL1841380 0.79 MTOR (0.60) ATRMTORKCNH2PIK3CARPTOR
SCHEMBL15190013 0.78 MTOR (0.57) MTORKCNH2PIK3CARPTORMLST8
SCHEMBL3260866 0.78 MTOR (0.57) MTORKCNH2PIK3CARPTORMLST8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318377-B1 PYRIMIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE GENENTECH INC (US) 2013-08-21 EP claimed
WO-2010014939-A1 PYRIMIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE GENENTECH, INC. (US) 2010-02-04 WO disclosed