SCHEMBL3235296

SCHEMBL3235296

Nc1cc(F)ccc1NC(=O)CCCCCC(=O)Nc1nc(-c2ccc(F)cc2)cs1

nearest known ligand 0.70

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 13/20 0.70
HDAC6 Q9UBN7 9/20 0.70
HDAC9 Q9UKV0 8/20 0.70
LMNA P02545 2/20 0.66
MAPK1 P28482 2/20 0.66
HDAC3 O15379 10/20 0.62
HDAC2 Q92769 8/20 0.62
HDAC10 Q969S8 8/20 0.62
NCOR2 Q9Y618 2/20 0.62
SMN1; SMN2 Q16637 1/20 0.59
KMT2A Q03164 3/20 0.57
HDAC8 Q9BY41 5/20 0.55
HDAC4 P56524 4/20 0.55
HDAC7 Q8WUI4 4/20 0.55
HDAC11 Q96DB2 4/20 0.55
HDAC5 Q9UQL6 4/20 0.55
MEN1 O00255 2/20 0.55
RAB9A P51151 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3238723 0.94 HDAC1 (0.61) HDAC1HDAC6HDAC9LMNAMAPK1
SCHEMBL3241203 0.92 HDAC1 (0.64) HDAC1HDAC6HDAC9LMNAMAPK1
SCHEMBL3228076 0.88 HDAC3 (0.55) HDAC1HDAC6HDAC9LMNAMAPK1
SCHEMBL3238457 0.85 HDAC1 (0.56) HDAC1HDAC6HDAC9HDAC3HDAC2
SCHEMBL3235298 0.84 HDAC1 (0.54) HDAC1HDAC6HDAC9LMNAMAPK1
SCHEMBL7924376 0.83 MAPK1 (0.93) HDAC1HDAC6HDAC9LMNAMAPK1
SCHEMBL3237865 0.83 HDAC3 (0.53) HDAC1HDAC6HDAC9LMNAMAPK1
SCHEMBL3242900 0.82 HDAC1 (0.65) HDAC1HDAC6HDAC9LMNAMAPK1
SCHEMBL7929398 0.80 HDAC1 (0.74) HDAC1HDAC6HDAC9HDAC3HDAC2
SCHEMBL3238257 0.79 HDAC3 (0.76) HDAC1HDAC6HDAC9HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO claimed
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed