Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL3235690

COc1cc(C)c(S(=O)(=O)N(Cc2cc(C(=O)N3CCN(CC(=O)Nc4cccnc4)CC3)co2)C2CC2)c(C)c1.COc1cc(C)c(S(=O)(=O)N(Cc2cc(C(=O)N3CCN(CCCN(C)C)CC3)co2)C2CC2)c(C)c1.O=C(O)C(F)(F)F

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 6/20 0.39
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
DRD2 P14416 2/20 0.34
DRD3 P35462 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
HPGD P15428 2/20 0.32
CYP11B2 P19099 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
USP2 O75604 1/20 0.32
MAPT P10636 1/20 0.32
SIGLEC9 Q9Y336 1/20 0.31
AVPR1B P47901 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL2237905 0.94 CHRNB4 (0.39) CHRNB4CHRNA3DRD2DRD3SMN1; SMN2
SCHEMBL12346740 0.90 CHRNB4 (0.42) CHRNB4CHRNA3DRD2DRD3SMN1; SMN2
Trifluoroacetic Acid SCHEMBL2239467 0.88 BDKRB1 (0.49) BDKRB1
SCHEMBL12346741 0.83 BDKRB1 (0.53) BDKRB1DRD2
Trifluoroacetic Acid SCHEMBL2237661 0.83 KDM4E (0.44) TDP1USP2MAPT
Trifluoroacetic Acid SCHEMBL2242040 0.82 BDKRB1 (0.40) BDKRB1DRD2CYP2D6TDP1MAPT
SCHEMBL2237908 0.81 TDP1 (0.34) BDKRB1DRD2DRD3HPGDCYP1A2
Trifluoroacetic Acid SCHEMBL2239201 0.81 THRB (0.40) BDKRB1DRD2DRD3CYP3A4CYP2C9
Trifluoroacetic Acid SCHEMBL2243351 0.80 BDKRB1 (0.39) BDKRB1DRD2TDP1MAPT
Trifluoroacetic Acid SCHEMBL2237417 0.80 BDKRB1 (0.38) BDKRB1CYP3A4TDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010020556-A1 NEW BRADYKININ B1 ANTAGONISTS EVOTEC NEUROSCIENCES GMBH (DE) 2010-02-25 WO claimed