SCHEMBL3237454

SCHEMBL3237454

O=C(O)Oc1cn(Cc2cc(C(F)(F)F)ccc2Cl)c2c(F)ccc(F)c2c1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.41
MRGPRX4 Q96LA9 3/20 0.37
PPARG P37231 2/20 0.36
P2RX7 Q99572 3/20 0.35
FFAR4 Q5NUL3 1/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.35
ALDH1A1 P00352 1/20 0.35
TRAP1 Q12931 2/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90B1 P14625 1/20 0.35
SCN1A P35498 1/20 0.34
SCN4A P35499 1/20 0.34
SCN7A Q01118 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
SCN2A Q99250 1/20 0.34
SCN3A Q9NY46 1/20 0.34
SCN8A Q9UQD0 1/20 0.34
KDM4E B2RXH2 1/20 0.33
FFAR1 O14842 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3238442 0.92 CHRM1 (0.41) CHRM1MRGPRX4P2RX7PTGDR2KDM4E
SCHEMBL3234599 0.87 CHRM1 (0.44) CHRM1MRGPRX4P2RX7ALDH1A1TRAP1
SCHEMBL3237430 0.86 CHRM1 (0.53) CHRM1MRGPRX4P2RX7ALDH1A1KDM4E
SCHEMBL2883187 0.85 CHRM1 (0.56) CHRM1MRGPRX4P2RX7ALDH1A1TRAP1
SCHEMBL3242122 0.82 CHRM1 (0.48) CHRM1P2RX7
SCHEMBL3242155 0.82 CHRM1 (0.45) CHRM1P2RX7ALDH1A1KDM4E
SCHEMBL3238772 0.80 CHRM1 (0.44) CHRM1PPARGP2RX7ALDH1A1KDM4E
SCHEMBL3234252 0.79 CHRM1 (0.44) CHRM1MRGPRX4P2RX7PTGDR2
SCHEMBL3239024 0.77 CHRM1 (0.57) CHRM1
SCHEMBL2877226 0.76 CHRM1 (0.57) CHRM1MRGPRX4P2RX7ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-B1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK SHARP & DOHME (US) 2010-07-28 EP claimed