SCHEMBL3239254

SCHEMBL3239254

NC(=O)OC1CCN(C2(Cc3cccc(Cl)c3)C(=O)Nc3cc(Cl)ccc32)CC1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 19/20 0.49
TP53 P04637 14/20 0.49
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3252191 0.89 MDM2 (0.53) MDM2TP53MEN1KMT2A
SCHEMBL1325239 0.88 MDM2 (0.51) MDM2TP53MEN1KMT2A
SCHEMBL3239157 0.87 MDM2 (0.49) MDM2TP53MEN1KMT2A
SCHEMBL1322322 0.85 MDM2 (0.52) MDM2TP53MEN1KMT2A
SCHEMBL1320307 0.82 MDM2 (0.52) MDM2TP53
SCHEMBL1319084 0.82 MDM2 (0.53) MDM2TP53MEN1KMT2A
SCHEMBL3241327 0.81 MDM2 (0.53) MDM2TP53MEN1KMT2A
SCHEMBL3970399 0.81 MDM2 (0.51) MDM2TP53
SCHEMBL1325985 0.81 MDM2 (0.55) MDM2TP53MEN1KMT2A
SCHEMBL1320230 0.80 MDM2 (0.49) MDM2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2066318-B1 OXINDOLE DERIVATIVES AS ANTICANCER AGENTS HOFFMANN LA ROCHE (CH) 2010-05-12 EP claimed