SCHEMBL3242977

SCHEMBL3242977

Cc1c(C(=O)O)c2cccc(F)c2c(=O)n1C(C)[C@H]1CCCN1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 8/20 0.34
SLC6A2 P23975 6/20 0.34
SLC6A4 P31645 4/20 0.34
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
DHFR P00374 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2836915 1.00 SLC6A3 (0.34) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL3236796 1.00 SLC6A3 (0.34) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL2831354 1.00 SLC6A3 (0.34) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL2149129 0.88 SLC6A3 (0.37) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL2149025 0.88 SLC6A3 (0.37) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL2837237 0.87 SLC6A2 (0.36) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL2829896 0.87 SLC6A2 (0.36) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL2837387 0.86 SLC6A2 (0.35) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL2834248 0.86 SLC6A2 (0.35) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL2834258 0.79 KDM4E (0.43) MEN1KMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028655-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-03-18 WO disclosed