SCHEMBL3243116

SCHEMBL3243116

COc1cccc(OC)c1-c1cnnc(Cl)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 5/20 0.49
HSP90AB1 P08238 3/20 0.49
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HTR7 P34969 1/20 0.38
NQO2 P16083 2/20 0.37
KDM4E B2RXH2 2/20 0.37
MAPT P10636 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
S1PR4 O95977 1/20 0.34
G6PD P11413 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3239822 0.91 HSP90AA1 (0.44) HSP90AA1HSP90AB1ALDH1A1KMT2AMEN1
SCHEMBL3249911 0.82 MAPT (0.57) ALDH1A1KMT2AMEN1L3MBTL1KDM4E
SCHEMBL3256327 0.81 PDE2A (0.38) HSP90AA1HSP90AB1ALDH1A1KMT2AMEN1
SCHEMBL3246149 0.80 HSP90AA1 (0.56) HSP90AA1HSP90AB1ALDH1A1HTR7KDM4E
SCHEMBL3257237 0.70 MAPT (0.41) HSP90AA1HSP90AB1HTR7KDM4EMAPT
SCHEMBL28668869 0.68 HSP90AA1 (0.50) HSP90AA1HSP90AB1ALDH1A1HTR7
SCHEMBL28148154 0.66 CA1 (0.65) ALDH1A1KMT2AMEN1L3MBTL1NQO2
SCHEMBL3244019 0.66 TLR8 (0.40) HSP90AA1HSP90AB1KMT2AMEN1KDM4E
SCHEMBL14450978 0.66 HSP90AA1 (0.44) HSP90AA1HSP90AB1ALDH1A1KMT2AMEN1
SCHEMBL9910949 0.66 CCR1 (0.58) HSP90AA1HSP90AB1HTR7NQO2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010001220-A1 NEW 1,2,4-TRIAZINE DERIVATIVES AND BIOLOGICAL APPLICATIONS THEREOF MUTABILIS SA (FR) 2010-01-07 WO disclosed
EP-2141164-A1 New 1,2,4-triazine derivatives and biological applications thereof Mutabilis (FR) 2010-01-06 EP disclosed