SCHEMBL3246149

SCHEMBL3246149

COc1cccc(OC)c1-c1cnnc(N)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 5/20 0.56
HSP90AB1 P08238 3/20 0.56
ADORA2A P29274 2/20 0.44
ADORA1 P30542 2/20 0.44
CHRNA7 P36544 1/20 0.42
DCPS Q96C86 1/20 0.41
MCHR1 Q99705 1/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
RAB9A P51151 1/20 0.39
TDP1 Q9NUW8 2/20 0.38
CYP3A4 P08684 1/20 0.38
HTR7 P34969 2/20 0.38
HTR1A P08908 1/20 0.38
HTR2B P41595 1/20 0.38
HTR5A P47898 1/20 0.38
NFATC1 O95644 1/20 0.38
GSK3B P49841 1/20 0.38
DYRK1A Q13627 1/20 0.38
ADRA2B P18089 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3393346 0.82 HSP90AA1 (0.59) HSP90AA1HSP90AB1ADORA2AADORA1CHRNA7
SCHEMBL13425400 0.81 GAA (0.50) HSP90AA1HSP90AB1ADORA2AADORA1ALDH1A1
SCHEMBL3243116 0.80 HSP90AA1 (0.49) HSP90AA1HSP90AB1ALDH1A1KDM4ERAB9A
SCHEMBL3398225 0.79 ADORA2A (0.49) HSP90AA1ADORA2AADORA1ALDH1A1HTR7
SCHEMBL3239822 0.75 HSP90AA1 (0.44) HSP90AA1HSP90AB1ALDH1A1KDM4ERAB9A
SCHEMBL3952084 0.75 HSP90AA1 (0.71) HSP90AA1HSP90AB1ADORA2AADORA1CHRNA7
SCHEMBL28668869 0.75 HSP90AA1 (0.50) HSP90AA1HSP90AB1CHRNA7DCPSMCHR1
SCHEMBL3952648 0.73 HSP90AA1 (0.81) HSP90AA1HSP90AB1CHRNA7DCPSALDH1A1
SCHEMBL2322961 0.73 ADORA2A (0.50) ADORA2AADORA1ALDH1A1KDM4ERAB9A
SCHEMBL6385078 0.72 KDM4E (0.49) ADORA2AADORA1ALDH1A1KDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010001220-A1 NEW 1,2,4-TRIAZINE DERIVATIVES AND BIOLOGICAL APPLICATIONS THEREOF MUTABILIS SA (FR) 2010-01-07 WO disclosed
EP-2141164-A1 New 1,2,4-triazine derivatives and biological applications thereof Mutabilis (FR) 2010-01-06 EP disclosed