SCHEMBL3243707

SCHEMBL3243707

O=C(O)NC1=CC(c2cccc(O)c2)(c2ccnc(C(F)(F)F)c2)Nc2cc[nH]c21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.34
OPRM1 P35372 1/20 0.33
OPRL1 P41146 1/20 0.33
MALT1 Q9UDY8 1/20 0.33
SMARCA2 P51531 1/20 0.31
SMARCA4 P51532 1/20 0.31
PRKD3 O94806 1/20 0.31
PRKCG P05129 1/20 0.31
CDK1 P06493 1/20 0.31
CDK2 P24941 1/20 0.31
FLT4 P35916 1/20 0.31
FLT3 P36888 1/20 0.31
FRK P42685 1/20 0.31
CDK8 P49336 1/20 0.31
CSNK2A1 P68400 1/20 0.31
CDK5 Q00535 1/20 0.31
ACVR1 Q04771 1/20 0.31
MST1R Q04912 1/20 0.31
STK3 Q13188 1/20 0.31
PTK6 Q13882 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3244253 0.69 BACE1 (0.40) HDAC4MALT1SMARCA2SMARCA4SYK
SCHEMBL3244258 0.66 HDAC4 (0.37) HDAC4OPRM1OPRL1SYK
SCHEMBL3616240 0.60 SMARCA2 (0.66) HDAC4MALT1SMARCA2SMARCA4
SCHEMBL3239041 0.58 BACE1 (0.36) OPRM1OPRL1SYK
SCHEMBL2463393 0.58 BACE1 (0.58)
SCHEMBL3239035 0.58 BACE1 (0.52) OPRM1OPRL1SYK
SCHEMBL29769017 0.57 LOXL2 (0.52) HDAC4SMARCA2SMARCA4SYK
SCHEMBL1199840 0.57 LOXL2 (0.52) HDAC4SMARCA2SMARCA4SYK
SCHEMBL31644090 0.56 SMARCA2 (0.42) HDAC4SMARCA2SMARCA4
SCHEMBL27597129 0.55 SYK (0.50) SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010056195-A1 NEW COMPOUNDS 575 ASTRAZENECA AB (SE) 2010-05-20 WO disclosed