SCHEMBL3244372

SCHEMBL3244372

CC(Oc1ccc(CC2SC(=O)NC2=O)cc1)c1nc2ccc(OCCc3ccc(N)cc3)cc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.47
PPARG P37231 12/20 0.47
CYP3A4 P08684 1/20 0.45
RXRA P19793 1/20 0.45
FFAR1 O14842 8/20 0.42
PPARA Q07869 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6544249 0.91 MAPT (0.50) MAPTPPARGFFAR1PPARA
Hydrochloric Acid SCHEMBL3243785 0.90 MAPT (0.49) MAPTPPARGCYP3A4RXRAFFAR1
SCHEMBL3251992 0.88 PPARG (0.45) MAPTPPARGCYP3A4RXRAFFAR1
Hydrochloric Acid SCHEMBL7121282 0.88 PPARG (0.42) MAPTPPARGCYP3A4RXRAFFAR1
Hydrochloric Acid SCHEMBL3246258 0.88 PPARG (0.44) MAPTPPARGCYP3A4RXRAFFAR1
SCHEMBL1130792 0.86 PPARG (0.54) PPARGFFAR1PPARA
Hydrochloric Acid SCHEMBL6064786 0.85 PPARG (0.53) PPARGCYP3A4RXRAFFAR1PPARA
Hydrochloric Acid SCHEMBL4165069 0.85 PPARG (0.53) PPARGCYP3A4RXRAFFAR1PPARA
SCHEMBL7241918 0.85 FFAR1 (0.54) PPARGFFAR1PPARA
Hydrochloric Acid SCHEMBL3240947 0.85 PPARG (0.45) MAPTPPARGFFAR1PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1167366-B1 AMINE DERIVATIVES DAIICHI SANKYO CO LTD (JP) 2010-05-05 EP disclosed
US-6562849-B1 Amine compound or pharmacologically acceptable salt thereof. These compounds are useful in the treatment and/or prophylaxis of diseases such as diabetes, hyperlipemia, arteriosclerosis, cancer, etc. SANKYO COMPANY, LIMITED (JP) 2003-05-13 US disclosed
US-20030078426-A1 Amine derivative compounds SANKYO COMPANY, LIMITED (JP) 2003-04-24 US disclosed
EP-1167366-A1 AMINE DERIVATIVES Sankyo Company, Limited (JP) 2002-01-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078426-A1 Amine derivative compounds H1-10, APOB, PRMT1 MAPT 4153/4885PPARG 929/4885CYP3A4 3494/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.