SCHEMBL3245010

SCHEMBL3245010

CCN(Cc1ccccc1)C(=O)Nc1ccc(-c2cn[nH]c2)cc1OC

nearest known ligand 0.70

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 20/20 0.70
ROCK1 Q13464 9/20 0.64
CDC42BPA Q5VT25 3/20 0.64
CYP3A4 P08684 2/20 0.52
CYP2D6 P10635 2/20 0.52
CYP2C9 P11712 2/20 0.52
AKT1 P31749 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13391088 0.92 ROCK2 (0.83) ROCK2ROCK1CDC42BPACYP3A4CYP2D6
SCHEMBL3240921 0.91 ROCK2 (0.81) ROCK2ROCK1CDC42BPACYP3A4CYP2D6
SCHEMBL3126886 0.88 ROCK2 (0.64) ROCK2ROCK1CDC42BPACYP2C9AKT1
SCHEMBL3239736 0.87 ROCK2 (0.92) ROCK2ROCK1CDC42BPACYP3A4CYP2D6
SCHEMBL13391314 0.85 ROCK2 (0.83) ROCK2ROCK1CDC42BPA
SCHEMBL3251485 0.85 ROCK2 (0.83) ROCK2ROCK1CDC42BPA
SCHEMBL3116361 0.85 ROCK2 (0.83) ROCK2ROCK1CDC42BPA
SCHEMBL3130458 0.84 ROCK2 (0.69) ROCK2ROCK1CDC42BPA
SCHEMBL13391372 0.83 ROCK2 (0.81) ROCK2ROCK1CDC42BPACYP3A4CYP2D6
SCHEMBL13391347 0.83 ROCK2 (0.88) ROCK2ROCK1CDC42BPACYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO claimed
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO disclosed