SCHEMBL3246979

SCHEMBL3246979

COc1ccc2c(c1)CN(C(=O)CN1C(=O)CCc3cc(-c4cc(Cl)ccn4)cnc31)CC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PORCN Q9H237 1/20 0.40
MAPK1 P28482 4/20 0.39
ESR2 Q92731 2/20 0.38
ESR1 P03372 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
ABCB1 P08183 1/20 0.37
ABCC1 P33527 1/20 0.37
MAPT P10636 2/20 0.37
HPGD P15428 2/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HSD17B3 P37058 2/20 0.37
CHRM4 P08173 1/20 0.36
SPR P35270 1/20 0.36
GRIN2C Q14957 1/20 0.36
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
POLB P06746 1/20 0.36
NR4A1 P22736 1/20 0.36
APEX1 P27695 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3128418 0.94 ROCK1 (0.37) PORCNMAPK1ESR2ESR1HSD17B3
SCHEMBL3243203 0.89 TAAR1 (0.43) PORCNESR2ESR1TAAR1ABCB1
SCHEMBL3264528 0.89 MAPK1 (0.44) PORCNMAPK1ESR2ESR1TAAR1
SCHEMBL3127545 0.89 MAPK1 (0.41) PORCNMAPK1ESR2ESR1TAAR1
SCHEMBL13521598 0.88 HSD17B3 (0.43) MAPK1ESR2ESR1TAAR1ABCB1
SCHEMBL3244932 0.88 TSHR (0.43) PORCNMAPK1ESR2TAAR1ABCB1
SCHEMBL3246260 0.86 CYP11B1 (0.48) PORCNMAPK1ESR2ESR1TAAR1
SCHEMBL3118590 0.85 ESR2 (0.45) MAPK1ESR2ESR1TAAR1ABCB1
SCHEMBL3119024 0.85 TAAR1 (0.46) PORCNMAPK1ESR2ESR1TAAR1
SCHEMBL3124617 0.85 GRIN2B (0.42) PORCNMAPK1ESR2ESR1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO claimed