SCHEMBL3264528

SCHEMBL3264528

COc1ccc2c(c1)CN(C(=O)CN1C(=O)CCc3cc(-c4ccc(Cl)cc4)cnc31)CC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 5/20 0.44
ABCB1 P08183 1/20 0.43
ABCC1 P33527 1/20 0.43
HSD17B3 P37058 2/20 0.42
ESR2 Q92731 2/20 0.41
ESR1 P03372 1/20 0.41
PORCN Q9H237 1/20 0.41
TAAR1 Q96RJ0 1/20 0.40
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 1/20 0.40
GRIN1 Q05586 2/20 0.39
GRIN2B Q13224 2/20 0.39
MAPT P10636 3/20 0.39
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
NR4A1 P22736 1/20 0.39
APEX1 P27695 1/20 0.39
RECQL P46063 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3127545 0.93 MAPK1 (0.41) MAPK1ABCB1ABCC1ESR2ESR1
SCHEMBL3119024 0.92 TAAR1 (0.46) MAPK1ABCB1ABCC1ESR2ESR1
SCHEMBL3124617 0.91 GRIN2B (0.42) MAPK1ABCB1ABCC1HSD17B3ESR2
SCHEMBL13521598 0.91 HSD17B3 (0.43) MAPK1ABCB1HSD17B3ESR2ESR1
SCHEMBL3246260 0.91 CYP11B1 (0.48) MAPK1ABCB1ABCC1ESR2ESR1
SCHEMBL3118590 0.90 ESR2 (0.45) MAPK1ABCB1ABCC1ESR2ESR1
SCHEMBL3248554 0.89 ESR2 (0.41) MAPK1ABCB1ABCC1ESR2ESR1
SCHEMBL13521725 0.89 CYP11B1 (0.47) MAPK1ABCB1HSD17B3ESR2ESR1
SCHEMBL3246979 0.89 PORCN (0.40) MAPK1ABCB1ABCC1HSD17B3ESR2
SCHEMBL13521603 0.88 MAPK1 (0.43) MAPK1ABCB1ESR2ESR1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed