SCHEMBL3247160

SCHEMBL3247160

CNc1ccc(Cl)cc1C1NCCc2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRCP P42785 5/20 0.57
GAA P10253 2/20 0.47
GID4 Q8IVV7 1/20 0.44
HTR2A P28223 4/20 0.43
HTR2C P28335 4/20 0.43
HTR2B P41595 4/20 0.43
ADRB1 P08588 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
CNR1 P21554 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
HRH1 P35367 1/20 0.43
KCNH2 Q12809 1/20 0.43
RECQL P46063 1/20 0.43
ALOX12 P18054 2/20 0.42
MAPT P10636 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cadaverine Tartrate SCHEMBL5873445 0.90 PRCP (0.47) PRCPGAAGID4ALOX12MAPT
SCHEMBL27893411 0.80 PRCP (0.63) PRCPGAAHTR2AHTR2CHTR2B
SCHEMBL8331546 0.75 FADS1 (0.36) PRCPGAAHTR2AHTR2CHTR2B
SCHEMBL14900840 0.74 PRCP (0.51) PRCPGAAGID4HTR2AHTR2C
SCHEMBL21063715 0.73 PRCP (1.00) PRCPGAAGID4RECQLOPRM1
SCHEMBL30973226 0.73 PRCP (1.00) PRCPGAAGID4RECQLOPRM1
SCHEMBL3072702 0.73 PRCP (1.00) PRCPGAAGID4RECQLOPRM1
SCHEMBL14677303 0.73 PRCP (0.65) PRCPGAAGID4HTR2AHTR2C
SCHEMBL22728767 0.73 PRCP (0.69) PRCPGAAGID4RECQLOPRM1
SCHEMBL28190726 0.73 PRCP (0.69) PRCPGAAGID4RECQLOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227803-B1 COMPOUNDS FOR INHIBITING IAPP-ASSOCIATED AMYLOID DEPOSITS BELLUS HEALTH INTERNATIONAL LTD (CH) 2010-05-05 EP claimed
US-6562836-B1 Islet amyloid polypeptide (IAPP) is known to be capable of forming fibrils which are deposited in the pancreas of patients wtih type II diabetes QUEEN'S UNIVERSITY OF KINGSTON (CA) 2003-05-13 US claimed
US-7393875-B2 Reducing islet amyloid polypeptide (IAPP) associated deposit; type II diabetes NEUROCHEM (INTERNATIONAL) LIMITED (CH) 2008-07-01 US disclosed
EP-1057814-B1 TETRAHYDROBENZINDOLE DERIVATIVES MEIJI SEIKA KAISHA (JP) 2005-03-09 EP disclosed
US-6498251-B1 Tetrahydrobenzindole derivatives MEIJI SEIKA KAISHA, LTD. (JP) 2002-12-24 US disclosed
EP-1057814-A1 TETRAHYDROBENZINDOLE DERIVATIVES Meiji Seika Kaisha, Ltd. (JP) 2000-12-06 EP disclosed