SCHEMBL3248337

SCHEMBL3248337

COC(=O)C1=C(C)Nc2nnnn2C1c1cccc2ccccc12

nearest known ligand 0.75

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.75
SMN1; SMN2 Q16637 3/20 0.67
HPGD P15428 3/20 0.62
HTT P42858 2/20 0.62
NPSR1 Q6W5P4 3/20 0.61
LMNA P02545 3/20 0.60
PKM P14618 1/20 0.59
MAPT P10636 2/20 0.57
TP53 P04637 1/20 0.55
KMT2A Q03164 3/20 0.55
THRB P10828 1/20 0.53
GAA P10253 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2996112 0.89 ALDH1A1 (0.76) ALDH1A1SMN1; SMN2HPGDHTTNPSR1
SCHEMBL3248182 0.89 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2HPGDHTTNPSR1
SCHEMBL3115427 0.88 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2HTTNPSR1LMNA
SCHEMBL13209867 0.86 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2HPGDHTTNPSR1
SCHEMBL3265207 0.86 ALDH1A1 (0.67) ALDH1A1SMN1; SMN2HTTNPSR1LMNA
SCHEMBL4263306 0.86 ALDH1A1 (0.77) ALDH1A1SMN1; SMN2HPGDHTTNPSR1
SCHEMBL3243075 0.85 MAPT (0.56) ALDH1A1SMN1; SMN2HPGDHTTNPSR1
SCHEMBL3223845 0.85 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2HPGDHTTNPSR1
SCHEMBL2996576 0.85 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2HPGDHTTNPSR1
SCHEMBL2999529 0.85 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2HPGDHTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010002483-A1 OPTIONALLY CONDENSED DIHYDRO PYRIDINE, DIHYDROPYRIMIDINE AND DIHYDRO PYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2010-01-07 WO disclosed
WO-2009006580-A1 OPTIONALLY CONDENSED DIHYDROPYRIDINE, DIHYDROPYRIMIDINE AND DIHYDROPYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2009-01-08 WO disclosed