SCHEMBL3248676

SCHEMBL3248676

COc1cccc(COC(=O)Nc2ccc(-c3cn[nH]c3)cc2OC2CCC(O)CC2)c1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 16/20 0.58
ROCK1 Q13464 4/20 0.58
CDC42BPA Q5VT25 4/20 0.58
PRKACA P17612 1/20 0.47
PRKACG P22612 1/20 0.47
PRKACB P22694 1/20 0.47
CYP2C9 P11712 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3244488 0.96 ROCK2 (0.57) ROCK2ROCK1CDC42BPAPRKACAPRKACG
SCHEMBL3252386 0.91 ROCK2 (0.57) ROCK2ROCK1CDC42BPACYP2C9NPC1
SCHEMBL3247404 0.88 ROCK2 (0.74) ROCK2ROCK1CDC42BPAPRKACAPRKACG
SCHEMBL3241016 0.88 ROCK2 (0.56) ROCK2ROCK1CDC42BPACYP2C9
SCHEMBL3241015 0.87 ROCK2 (0.63) ROCK2ROCK1CDC42BPAPRKACAPRKACG
SCHEMBL3241104 0.83 ROCK2 (0.62) ROCK2ROCK1CDC42BPAPRKACAPRKACG
SCHEMBL3248264 0.83 ROCK2 (0.62) ROCK2ROCK1CDC42BPAPRKACAPRKACG
SCHEMBL3240773 0.83 ROCK2 (0.52) ROCK2ROCK1CDC42BPAPRKACAPRKACG
SCHEMBL3253611 0.82 ROCK2 (0.61) ROCK2ROCK1CDC42BPACYP2C9NPC1
SCHEMBL3247408 0.82 ROCK2 (0.68) ROCK2ROCK1CDC42BPACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO claimed
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO disclosed