SCHEMBL3249992

SCHEMBL3249992

CCCN1CCc2c([nH]c3ccccc23)C1CC(=O)O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.56
ABCG2 Q9UNQ0 3/20 0.53
ABCB1 P08183 2/20 0.53
KDM4E B2RXH2 4/20 0.50
PGR P06401 1/20 0.49
TUBB4A P04350 1/20 0.48
TUBB P07437 1/20 0.48
TUBA3C P0DPH7 1/20 0.48
TUBA1B P68363 1/20 0.48
TUBA4A P68366 1/20 0.48
TUBB4B P68371 1/20 0.48
TUBB3 Q13509 1/20 0.48
TUBB2A Q13885 1/20 0.48
TUBB8 Q3ZCM7 1/20 0.48
TUBA3E Q6PEY2 1/20 0.48
TUBA1A Q71U36 1/20 0.48
TUBA1C Q9BQE3 1/20 0.48
TUBB6 Q9BUF5 1/20 0.48
TUBB2B Q9BVA1 1/20 0.48
TUBB1 Q9H4B7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3240544 0.85 ESR1 (0.54) ESR1ABCG2ABCB1KDM4EPGR
SCHEMBL16373146 0.79 SIGMAR1 (0.71) ESR1ABCG2ABCB1KDM4EPGR
SCHEMBL11479762 0.78 ESR1 (0.54) ESR1ABCG2ABCB1KDM4EMEN1
Hydrochloric Acid SCHEMBL11472041 0.77 ESR1 (0.53) ESR1ABCG2ABCB1KDM4EMEN1
SCHEMBL11176271 0.74 KDM4E (0.48) ESR1ABCG2ABCB1KDM4EMEN1
SCHEMBL11481659 0.74 KDM4E (0.48) ESR1ABCG2ABCB1KDM4EMEN1
Hydrochloric Acid SCHEMBL11470335 0.74 MEN1 (0.53) ESR1ABCG2ABCB1KDM4EMEN1
SCHEMBL11178936 0.74 KDM4E (0.47) ESR1ABCG2ABCB1KDM4EMEN1
SCHEMBL8386930 0.73 ESR1 (0.68) ESR1ABCG2ABCB1PGRLMNA
SCHEMBL11454881 0.73 MAPKAPK2 (0.50) ESR1ABCG2ABCB1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2102204-B1 NEW AMINOPYRROLO[1,2- A]INDOLE ET AMINOPYRIDAZINO[1,6-A]INDOLE DERIVATIVES, METHOD FOR PREPARING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SERVIER LAB (FR) 2010-05-05 EP disclosed