SCHEMBL3250242

SCHEMBL3250242

COc1cc2c(cc1OC)C(CCCC1c3cc(OC)c(OC)cc3CCN1C)N(C)CC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN2 Q9H2S1 4/20 1.00
KCNN3 Q9UGI6 4/20 1.00
KCNN1 Q92952 2/20 1.00
LMNA P02545 2/20 0.67
KDM4E B2RXH2 2/20 0.67
ALDH1A1 P00352 2/20 0.67
HSD17B10 Q99714 2/20 0.67
MAOA P21397 2/20 0.67
MAPK1 P28482 1/20 0.67
NR1I2 O75469 1/20 0.67
PTGS2 P35354 1/20 0.67
OPRK1 P41145 1/20 0.67
SLC6A3 Q01959 1/20 0.67
CYP2D6 P10635 1/20 0.67
ALOX15 P16050 1/20 0.62
GRIN2D O15399 5/20 0.57
GRIN3B O60391 5/20 0.57
GRIN1 Q05586 5/20 0.57
GRIN2A Q12879 5/20 0.57
GRIN2B Q13224 5/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3254146 0.98 KCNN2 (1.00) KCNN2KCNN3KCNN1LMNAKDM4E
SCHEMBL3253219 0.97 KCNN2 (0.94) KCNN2KCNN3KCNN1LMNAKDM4E
Hydrochloric Acid SCHEMBL3248635 0.95 KCNN2 (0.94) KCNN2KCNN3KCNN1LMNAKDM4E
SCHEMBL3251892 0.95 KCNN2 (0.91) KCNN2KCNN3KCNN1LMNAKDM4E
Hydrochloric Acid SCHEMBL5136925 0.94 KCNN2 (0.92) KCNN2KCNN3KCNN1LMNAKDM4E
Hydrochloric Acid SCHEMBL3250094 0.94 KCNN2 (0.92) KCNN2KCNN3KCNN1LMNAKDM4E
SCHEMBL13878183 0.86 KCNN2 (0.76) KCNN2KCNN3KCNN1LMNAKDM4E
SCHEMBL27961570 0.84 MAOA (0.72) KCNN2KCNN3KCNN1LMNAKDM4E
Hydrochloric Acid SCHEMBL10637118 0.83 KCNN2 (0.72) KCNN2KCNN3KCNN1LMNAKDM4E
SCHEMBL10642034 0.83 KCNN2 (0.70) KCNN2KCNN3KCNN1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1998775-B1 BIS1,2,3,4-TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR USES AS PHARMACEUTICALS UNIV LIEGE (BE) 2010-05-19 EP claimed