SCHEMBL3250792

SCHEMBL3250792

COc1ccc2c(c1)CC(S(=O)(=O)CCN(C)C)Cn1c-2c(C2CCCCC2)c2ccc(C(=O)O)cc21

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.52
MMP12 P39900 1/20 0.52
NR1I2 O75469 8/20 0.45
KCNH2 Q12809 7/20 0.45
CYP3A4 P08684 3/20 0.45
SCN5A Q14524 2/20 0.45
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
SCN9A Q15858 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14009712 0.93 NR1I2 (0.46) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL14009597 0.90 KCNH2 (0.57) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL14009657 0.83 KCNH2 (0.44) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL3943346 0.83 PRKCA (0.46) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL895975 0.81 PRKCA (0.49) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL5528023 0.80 PRKCA (0.47) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL14009596 0.80 NR1I2 (0.58) NR1I2KCNH2CYP3A4SCN5ACYP2C9
SCHEMBL2277325 0.80 PRKCA (0.46) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL894723 0.80 PRKCA (0.48) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL5002450 0.80 PRKCA (0.54) PRKCAMMP12NR1I2KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029606-B1 CYCLOPROPYL FUSED INDOLOBENZAZEPINE HCV NS5B INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2010-05-26 EP disclosed