SCHEMBL3253575

SCHEMBL3253575

COc1ccc(CCNc2nc(N3CCCC3CO)nc3ccccc23)cc1.OCC1CCCN1c1nc(NCCc2ccc(Br)cc2)c2ccccc2n1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 7/20 0.48
HRH4 Q9H3N8 1/20 0.47
CCNE2 O96020 1/20 0.46
CCNE1 P24864 1/20 0.46
CDK2 P24941 1/20 0.46
CCR4 P51679 1/20 0.44
ACP1 P24666 2/20 0.44
ACVR1 Q04771 1/20 0.43
APP P05067 1/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
HTR2A P28223 1/20 0.42
SLC2A1 P11166 1/20 0.42
PDE5A O76074 1/20 0.41
CDK5 Q00535 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2846271 0.96 CDK1 (0.51) CDK1HRH4CCNE2CCNE1CDK2
SCHEMBL2852678 0.93 HRH4 (0.51) CDK1HRH4CCNE2CCNE1CDK2
SCHEMBL13356604 0.88 HRH4 (0.52) HRH4ACP1APPBCHEACHE
SCHEMBL20733814 0.86 HRH4 (0.58) CDK1HRH4CCNE2CCNE1CDK2
SCHEMBL20718973 0.86 HRH4 (0.58) CDK1HRH4CCNE2CCNE1CDK2
SCHEMBL2845074 0.86 HRH4 (0.53) CDK1HRH4CCNE2CCNE1CDK2
SCHEMBL20718970 0.84 CCNE2 (0.62) CDK1HRH4CCNE2CCNE1CDK2
SCHEMBL20733875 0.84 HRH4 (0.57) CDK1HRH4CCNE2CCNE1CDK2
SCHEMBL3642691 0.78 HRH4 (0.66) HRH4ACP1APPHTR2ASLC2A1
Hydrochloric Acid SCHEMBL3641028 0.77 HRH4 (0.65) HRH4ACP1HTR2ASLC2A1PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010056907-A2 COMPOUNDS THAT INDUCE PANCREATIC BETA-CELL EXPANSION THE SCRIPPS RESEARCH INSTITUTE (US) 2010-05-20 WO claimed