SCHEMBL3254396

SCHEMBL3254396

Fc1ccc(Nc2ccc3c(C4=COC(c5ccccc5Cl)O4)n[nH]c3n2)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
NFKB1 P19838 1/20 0.39
RAB9A P51151 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAPK14 Q16539 9/20 0.38
MAPK9 P45984 1/20 0.32
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3251323 0.79 MAPK14 (0.48) KDM4ENPC1ALDH1A1GAANFKB1
SCHEMBL3254392 0.72 MAPK14 (0.41) KDM4ENPC1ALDH1A1GAANFKB1
SCHEMBL3251929 0.70 MAPK14 (0.47) KDM4ENPC1ALDH1A1GAANFKB1
SCHEMBL3249327 0.70 MAPK9 (0.51) KDM4ENPC1ALDH1A1GAANFKB1
SCHEMBL3253883 0.69 MAPK9 (0.47) KDM4ENPC1ALDH1A1GAANFKB1
SCHEMBL12467808 0.68 KDM4E (0.51) KDM4ENPC1ALDH1A1GAANFKB1
SCHEMBL3248737 0.66 KDM4E (0.41) KDM4ENPC1ALDH1A1GAANFKB1
SCHEMBL3252473 0.64 GSK3A (0.40) MAPK14MAPK9
SCHEMBL3250649 0.64 MAPK9 (0.47) NPC1RAB9ASMN1; SMN2MAPK14MAPK9
SCHEMBL13678697 0.62 MAPK9 (0.49) MAPK14MAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833477-B1 PYRAZOLO-HETEROARYL COMPOUNDS USEFUL TO TREAT TNF-ALPHA AND IL-1 MEDIATED DISEASES NOVARTIS AG (CH) 2010-06-02 EP claimed