SCHEMBL3256703

SCHEMBL3256703

CC1(C)CC(=C(c2ccc(F)cc2)c2ccc(C3=CCOC3=O)cc2)CC(C)(C)C1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.32
RARA P10276 1/20 0.31
RARB P10826 1/20 0.31
RARG P13631 1/20 0.31
SIGMAR1 Q99720 2/20 0.31
PTGS1 P23219 2/20 0.31
PTGS2 P35354 1/20 0.31
PDE3B Q13370 2/20 0.31
PDE3A Q14432 2/20 0.31
ESR1 P03372 1/20 0.30
DRD2 P14416 1/20 0.30
ALPL P05186 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6602632 0.77 PTGS1 (0.43) ALDH1A1SIGMAR1PTGS1PTGS2PDE3B
SCHEMBL6533645 0.76 HTR2A (0.39) ALDH1A1ESR1DRD2
SCHEMBL4620312 0.75 ESR1 (0.38) ALDH1A1PTGS1PTGS2ESR1
SCHEMBL3069374 0.74 LPL (0.39) ALDH1A1
SCHEMBL3074106 0.74 BCL2L1 (0.49) ALDH1A1RARARARBRARGESR1
SCHEMBL3068540 0.73 ESR1 (0.49) ALDH1A1PTGS1PTGS2ESR1
SCHEMBL3082420 0.73 LPL (0.38) ALDH1A1PTGS1PTGS2ESR1
SCHEMBL3133913 0.71 ESR1 (0.34) ALDH1A1ESR1
SCHEMBL3072806 0.69 BRD4 (0.48) PTGS1PTGS2
SCHEMBL3135618 0.69 ESR1 (0.54) ALDH1A1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891026-B1 CYCLOALKYLIDENE COMPOUNDS AS SELECTIVE ESTROGEN RECEPTOR MODULATORS GLAXOSMITHKLINE LLC (US) 2010-07-14 EP claimed