SCHEMBL325784

SCHEMBL325784

O=C(O)C1CN(C(=O)O)CC1c1cccc(Br)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.45
KDM1A O60341 2/20 0.44
HDAC4 P56524 1/20 0.43
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
GRK2 P25098 1/20 0.40
CASP6 P55212 1/20 0.40
CASP8 Q14790 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
PDE4B Q07343 2/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
TLR2 O60603 3/20 0.38
TLR1 Q15399 3/20 0.38
PPARG P37231 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015787 0.89 HRH3 (0.44) HRH3KDM1AHDAC4SLC6A4SLC6A3
SCHEMBL29900799 0.83 TLR2 (0.48) HRH3HDAC4ALDH1A1TLR2TLR1
SCHEMBL10311101 0.83 MEN1 (0.48) HRH3KDM1AHDAC4SLC6A4SLC6A3
SCHEMBL4342266 0.83 ALDH1A1 (0.40) TDP1HTR2AHTR2CHTR2BPDE4B
SCHEMBL15054630 0.83 ALDH1A1 (0.40) TDP1HTR2AHTR2CHTR2BPDE4B
SCHEMBL10277792 0.82 PDE4B (0.57) SLC6A4SLC6A3PDE4BPPARGPPARA
SCHEMBL10277788 0.82 PDE4B (0.57) SLC6A4SLC6A3PDE4BPPARGPPARA
SCHEMBL10277789 0.82 PDE4B (0.57) SLC6A4SLC6A3PDE4BPPARGPPARA
SCHEMBL528422 0.79 PDE4B (0.41) HRH3KDM1AHDAC4SLC6A4SLC6A3
SCHEMBL528421 0.79 PDE4B (0.41) HRH3KDM1AHDAC4SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590942-A1 RHO KINASE INHIBITORS Boehringer Ingelheim International GmbH (DE) 2013-05-15 EP disclosed
WO-2012006202-A1 RHO KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-12 WO disclosed