SCHEMBL3259676

SCHEMBL3259676

CNC(=O)c1cc2c(C)cccc2n(C(C)C)c1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 3/20 0.50
GLA P06280 3/20 0.50
GAA P10253 3/20 0.50
HPGD P15428 3/20 0.50
CASP1 P29466 3/20 0.50
CASP7 P55210 3/20 0.50
HSD17B10 Q99714 3/20 0.50
POLB P06746 2/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43
HTR4 Q13639 8/20 0.43
PKM P14618 1/20 0.43
HTT P42858 1/20 0.42
NPY5R Q15761 2/20 0.41
EZH2 Q15910 2/20 0.40
BRD4 O60885 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2010294 0.85 POLB (0.46) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL2010893 0.80 KDM4E (0.53) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL2008627 0.77 HTR4 (0.74) HTR4
SCHEMBL12572553 0.77 HTR4 (0.57) HTR4
Hydrochloric Acid SCHEMBL2006214 0.77 HTR4 (0.72) HTR4
SCHEMBL2012658 0.76 HTR4 (0.55) HTR4
SCHEMBL2006462 0.74 HTR4 (0.54) HTR4
SCHEMBL8287322 0.74 HTR4 (0.53) HTR4
Hydrochloric Acid SCHEMBL2009356 0.74 HTR4 (0.53) HTR4
SCHEMBL12630140 0.73 HTR4 (0.52) CYP3A4HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689742-B1 QUINOLONECARBOXYLIC ACID COMPOUNDS HAVING 5-HT4 RECEPTOR AGONISTIC ACTIVITY PFIZER (US) 2010-03-17 EP disclosed