SCHEMBL3260403

SCHEMBL3260403

CCOC(=O)c1cn(-c2ccccc2)nc1OCC

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.62
MAPK1 P28482 1/20 0.62
NPC1 O15118 4/20 0.60
RAB9A P51151 3/20 0.60
ALDH1A1 P00352 4/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
GLA P06280 1/20 0.55
NFKB1 P19838 1/20 0.55
NFKB2 Q00653 1/20 0.55
RELA Q04206 1/20 0.55
CA12 O43570 1/20 0.54
CA9 Q16790 1/20 0.54
POLB P06746 1/20 0.52
DGAT1 O75907 1/20 0.50
MAPT P10636 4/20 0.49
CHEK1 O14757 1/20 0.49
EGFR P00533 1/20 0.49
KDR P35968 1/20 0.49
HPGD P15428 2/20 0.49
TSHR P16473 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL720149 0.90 NPSR1 (0.58) NPSR1MAPK1NPC1RAB9AALDH1A1
SCHEMBL4291837 0.89 NPSR1 (0.62) NPSR1MAPK1NPC1RAB9AALDH1A1
SCHEMBL3260509 0.87 L3MBTL1 (0.51) NPSR1MAPK1NPC1RAB9AALDH1A1
SCHEMBL6172144 0.85 NPSR1 (0.67) NPSR1MAPK1NPC1RAB9AALDH1A1
SCHEMBL4854443 0.83 NPC1 (0.67) NPSR1MAPK1NPC1RAB9AALDH1A1
SCHEMBL2079861 0.82 NPSR1 (0.64) NPSR1MAPK1NPC1RAB9AALDH1A1
SCHEMBL22209257 0.82 NPSR1 (0.64) NPSR1MAPK1NPC1RAB9AALDH1A1
SCHEMBL20028758 0.82 NPSR1 (0.64) NPSR1MAPK1NPC1RAB9AALDH1A1
SCHEMBL22331103 0.81 NPSR1 (0.86) NPSR1MAPK1NPC1RAB9AALDH1A1
SCHEMBL20028759 0.81 NPSR1 (0.59) NPSR1MAPK1NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010015656-A2 NEW ALKOXYPYRAZOLES INSTITUT PASTEUR (FR) 2010-02-11 WO disclosed
WO-2010015656-A2 NEW ALKOXYPYRAZOLES INSTITUT PASTEUR (FR) 2010-02-11 WO disclosed
EP-2151434-A1 Alkoxypyrazoles and the process for their preparation Institut Pasteur (FR) 2010-02-10 EP disclosed
EP-2151434-A1 Alkoxypyrazoles and the process for their preparation Institut Pasteur (FR) 2010-02-10 EP disclosed