SCHEMBL3262928

SCHEMBL3262928

CS(=O)(=O)NCCOc1cccc(CN(CCO)C(=O)c2nc3ccc(-c4cn[nH]c4)cc3s2)c1

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 18/20 0.68
ROCK1 Q13464 8/20 0.66
CDC42BPA Q5VT25 4/20 0.66
MAPK10 P53779 1/20 0.66
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
CYP2C9 P11712 2/20 0.48
LCK P06239 1/20 0.43
ITK Q08881 1/20 0.43
PRKACA P17612 1/20 0.43
PRKACG P22612 1/20 0.43
PRKACB P22694 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13457432 0.90 ROCK2 (0.70) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL3265194 0.89 ROCK2 (0.78) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL3261889 0.88 ROCK2 (0.71) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL13457522 0.86 ROCK2 (0.86) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL13457384 0.86 ROCK2 (0.68) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL3260236 0.84 ROCK2 (0.66) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL13457050 0.82 ROCK2 (0.84) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL3251667 0.81 ROCK2 (0.73) ROCK2ROCK1CDC42BPACYP3A4CYP2D6
SCHEMBL13457123 0.81 ROCK2 (1.00) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL13457098 0.80 ROCK2 (1.00) ROCK2ROCK1CDC42BPAMAPK10CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010024903-A1 BENZO[d]OXAZOLES AND BENZO[d]THIAZOLES AS KINASE INHIBITORS FENG YANGBO (US) 2010-03-04 WO disclosed