SCHEMBL3264764

SCHEMBL3264764

CC1(C)OB(c2ccc(CN3CCC(F)CC3)c(F)c2)OC1(C)C

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.52
CXCR3 P49682 14/20 0.40
ALDH1A1 P00352 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
KDM4E B2RXH2 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LPL P06858 1/20 0.38
LIPG Q9Y5X9 1/20 0.38
CYP2A13 Q16696 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3263594 0.93 ROCK1 (0.50) ROCK1CXCR3ALDH1A1TDP1KDM4E
SCHEMBL3263593 0.93 ROCK1 (0.50) ROCK1CXCR3ALDH1A1TDP1KDM4E
SCHEMBL428922 0.89 CYP2A13 (0.50) ROCK1ALDH1A1KDM4ESMN1; SMN2LPL
SCHEMBL19211744 0.88 KDM4E (0.52) ROCK1CXCR3ALDH1A1KDM4ESMN1; SMN2
SCHEMBL18580506 0.88 ROCK1 (0.48) ROCK1CXCR3ALDH1A1TDP1KDM4E
SCHEMBL18580183 0.87 ROCK1 (0.45) ROCK1CXCR3ALDH1A1TDP1KDM4E
SCHEMBL21644162 0.87 KDM4E (0.55) ROCK1CXCR3ALDH1A1KDM4ESMN1; SMN2
SCHEMBL18579955 0.86 ROCK1 (0.53) ROCK1ALDH1A1TDP1KDM4ESMN1; SMN2
SCHEMBL2563557 0.86 ROCK1 (0.48) ROCK1CXCR3ALDH1A1TDP1KDM4E
SCHEMBL20198185 0.85 ROCK1 (0.49) ROCK1CXCR3ALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010010184-A1 [1, 2, 4] TRIAZOLO [1, 5-A] PYRIDINES AS JAK INHIBITORS GALAPAGOS NV (BE) 2010-01-28 WO disclosed