SCHEMBL3264966

SCHEMBL3264966

CCN(CC)CCNCCCNc1nnc2c(n1)c(=O)n(C)c(=O)n2C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
EGFR P00533 1/20 0.37
FGFR1 P11362 1/20 0.37
SRC P12931 1/20 0.37
FGFR2 P21802 1/20 0.37
FGFR4 P22455 1/20 0.37
FGFR3 P22607 1/20 0.37
CYP2D6 P10635 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
BLM P54132 1/20 0.36
CYP2C19 P33261 1/20 0.35
HTT P42858 4/20 0.35
GAA P10253 2/20 0.35
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34
KDM4E B2RXH2 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2183306 0.94 TP53 (0.41) TP53EGFRFGFR1SRCFGFR2
SCHEMBL2181684 0.92 FGFR1 (0.42) TP53EGFRFGFR1SRCFGFR2
SCHEMBL2183395 0.92 TP53 (0.47) TP53EGFRFGFR1SRCFGFR2
SCHEMBL2180532 0.85 CCND1 (0.35) TP53EGFRFGFR1SRCFGFR2
SCHEMBL2182521 0.83 LMNA (0.40) CYP2C19HTTADORA2BKDM4ELMNA
SCHEMBL2181859 0.83 TSHR (0.36) TP53EGFRFGFR1SRCFGFR2
SCHEMBL2181675 0.82 CYP2D6 (0.49) CYP2D6POLBMAPTTHRBBLM
SCHEMBL2183080 0.82 CYP2D6 (0.48) CYP2D6POLBCYP2C19HTTGAA
SCHEMBL2181496 0.82 CYP2C19 (0.40) CYP2D6POLBMAPTTHRBBLM
SCHEMBL2183519 0.80 TP53 (0.41) TP53CYP2D6POLBMAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010014798-A2 PYRIMIDOTRIAZINEDIONES AND PYRIMIDOPYRIMIDINEDIONES AND METHODS OF USING THE SAME THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2010-02-04 WO disclosed