SCHEMBL326606

SCHEMBL326606

O=C(O)c1nnc(-c2ccc(Cl)cc2)o1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.72
SMPD1 P17405 1/20 0.67
RAB9A P51151 3/20 0.61
SMN1; SMN2 Q16637 3/20 0.61
ALDH1A1 P00352 2/20 0.61
LMNA P02545 2/20 0.59
MAPK1 P28482 1/20 0.59
POLB P06746 1/20 0.56
KDM4E B2RXH2 3/20 0.53
NPC1 O15118 2/20 0.53
HSD17B10 Q99714 2/20 0.53
NOTUM Q6P988 1/20 0.53
TP53 P04637 1/20 0.53
TSHR P16473 1/20 0.53
PTGS2 P35354 2/20 0.51
MAOA P21397 1/20 0.50
MAOB P27338 1/20 0.50
ALOX15 P16050 1/20 0.49
ALOX12 P18054 1/20 0.49
CXCR5 P32302 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17377393 0.98 PTPN1 (0.70) PTPN1SMPD1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL27851472 0.87 MAPK1 (0.69) PTPN1SMPD1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL3823166 0.84 SMPD1 (0.65) PTPN1SMPD1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL2330752 0.83 PTPN1 (0.93) PTPN1RAB9ASMN1; SMN2ALDH1A1POLB
Lithium Ion SCHEMBL17377391 0.83 SMPD1 (0.63) PTPN1SMPD1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL30578677 0.82 PTPN1 (0.72) PTPN1SMPD1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL19075480 0.82 PTPN1 (0.72) PTPN1SMPD1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL8840165 0.82 PTPN1 (0.72) PTPN1RAB9ASMN1; SMN2ALDH1A1LMNA
SCHEMBL12171897 0.82 NPC1 (0.74) SMPD1RAB9ASMN1; SMN2LMNAMAPK1
Hydrochloric Acid SCHEMBL19118776 0.81 PTPN1 (0.89) PTPN1RAB9ASMN1; SMN2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4727549-A2 PLASMODIUM FALCIPARUM BLOOD STAGE INHIBITORS University of Georgia Research Foundation, Inc. (US) 2026-04-22 EP disclosed
US-20260097046-A1 PLASMODIUM FALCIPARUM BLOOD STAGE INHIBITORS UNIV GEORGIA (US) 2026-04-09 US disclosed
WO-2024258900-A2 PLASMODIUM FALCIPARUM BLOOD STAGE INHIBITORS UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 2024-12-19 WO disclosed
WO-2023231948-A1 ISR INHIBITORS, METHOD FOR PREPARING SAME, AND USE THEREOF 中国药科大学 2023-12-07 WO disclosed
CN-116768877-A ISR inhibitor and preparation method and application thereof 中国药科大学 2023-09-19 CN disclosed
EP-2590969-B1 Therapeutic agents 976 ASTRAZENECA AB (SE) 2014-10-15 EP disclosed
EP-2468717-B1 Heterocyclic Amide Compounds Useful as Kinase Inhibitors BRISTOL MYERS SQUIBB CO (US) 2013-11-20 EP disclosed
US-8546375-B2 (3-(4-(aminomethyl)phenoxy or phenylthio)azetidin-1-yl)(5-phenyl-1,3,4-oxadiazol-2-yl)methanone compounds ASTRAZENECA AB (SE) 2013-10-01 US disclosed
EP-2590969-A2 THERAPEUTIC AGENTS 976 AstraZeneca AB (SE) 2013-05-15 EP disclosed
US-8404689-B2 Heterocyclic amide compounds useful as kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2013-03-26 US disclosed
US-20080171741-A1 HETEROCYCLIC AMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2008-07-17 US disclosed
US-20080171741-A1 HETEROCYCLIC AMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2008-07-17 US disclosed
US-20080171741-A1 HETEROCYCLIC AMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2008-07-17 US disclosed
WO-2008057775-A2 HETEROCYCLIC AMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-15 WO disclosed
US-5888941-A Carbozamides with antifungal activity J. URIACH & CIA. S.A. (ES) 1999-03-30 US disclosed
EP-0783502-A1 NEW CARBOXAMIDES WITH ANTIFUNGAL ACTIVITY J. URIACH & CIA. S.A. (ES) 1997-07-16 EP disclosed
WO-1997005131-A1 NEW CARBOXAMIDES WITH ANTIFUNGAL ACTIVITY J. URIACH & CIA. S.A. (ES) 1997-02-13 WO disclosed
US-5591695-A Herbicidal [1,3,4]oxadiazoles and thiadiazoles AMERICAN CYANAMID CO. (US) 1997-01-07 US disclosed
CN-1134935-A Herbicidal (1,3,4) oxadiazoles and thiadiazoles AMERICAN CYANAMID CO (US) 1996-11-06 CN disclosed
EP-0726263-A2 Herbicidal (1,3,4)oxadiazoles and thiadiazoles American Cyanamid Company (US) 1996-08-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080171741-A1 HETEROCYCLIC AMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS MAP3K1, MAP3K8, MAP3K20 PTPN1 1195/4885SMPD1 982/4885RAB9A 796/4885
US-20260097046-A1 PLASMODIUM FALCIPARUM BLOOD STAGE INHIBITORS SUB1, PFN1, HCCS PTPN1 3027/4885SMPD1 966/4885RAB9A 1834/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.