SCHEMBL3266400

SCHEMBL3266400

N#CCC(=O)N1CCCc2ccc(C(F)(F)F)cc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XIAP P98170 1/20 0.48
BIRC2 Q13490 1/20 0.48
CNR2 P34972 1/20 0.46
KDM4E B2RXH2 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
NOTUM Q6P988 1/20 0.45
LMNA P02545 1/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43
MAPK1 P28482 1/20 0.43
RAB9A P51151 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ROCK1 Q13464 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
KCNJ2 P63252 1/20 0.41
BRD4 O60885 1/20 0.41
ATAD2 Q6PL18 1/20 0.41
HDAC3 O15379 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27544652 0.80 CNR2 (0.53) XIAPBIRC2CNR2SMN1; SMN2NOTUM
SCHEMBL9393577 0.79 CNR2 (0.52) XIAPBIRC2CNR2SMN1; SMN2NOTUM
SCHEMBL10241674 0.79 NOTUM (0.66) XIAPBIRC2CNR2SMN1; SMN2NOTUM
SCHEMBL2087233 0.78 SMN1; SMN2 (0.62) KDM4ESMN1; SMN2NOTUMMAPK1ALDH1A1
SCHEMBL7830913 0.77 CNR2 (0.47) XIAPBIRC2CNR2KDM4ESMN1; SMN2
SCHEMBL3653813 0.76 NOTUM (0.61) XIAPBIRC2KDM4ESMN1; SMN2NOTUM
SCHEMBL23207270 0.76 XIAP (0.58) XIAPBIRC2CNR2SMN1; SMN2NOTUM
SCHEMBL8893534 0.76 XIAP (0.58) XIAPBIRC2CNR2NOTUMNPC1
SCHEMBL7552151 0.72 NOTUM (0.63) KDM4ESMN1; SMN2NOTUMLMNARAB9A
SCHEMBL2530222 0.72 CNR2 (0.62) XIAPBIRC2CNR2NOTUMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740171-B1 INDOL-1-YL-ACETIC ACID DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-06-09 EP disclosed