SCHEMBL3266738

SCHEMBL3266738

CC(C)(C)OC(=O)N1C2CCC1CC(Oc1ccc3[nH]c(C(=O)O)cc3c1)C2

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 9/20 0.46
KMT2A Q03164 1/20 0.45
CHRM2 P08172 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
GPR119 Q8TDV5 3/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
SRD5A2 P31213 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PIN1 Q13526 1/20 0.41
AKR1C3 P42330 1/20 0.41
PDGFRB P09619 1/20 0.39
PDGFRA P16234 1/20 0.39
SMAD3 P84022 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3251118 1.00 HRH3 (0.46) HRH3KMT2ACHRM2CHRM1CHRM3
SCHEMBL3251113 1.00 HRH3 (0.46) HRH3KMT2ACHRM2CHRM1CHRM3
SCHEMBL3243609 1.00 HRH3 (0.46) HRH3KMT2ACHRM2CHRM1CHRM3
SCHEMBL3243608 1.00 HRH3 (0.46) HRH3KMT2ACHRM2CHRM1CHRM3
SCHEMBL3249504 0.88 KDM4E (0.53) HRH3KMT2AKDM4EALDH1A1HPGD
SCHEMBL3249499 0.88 KDM4E (0.53) HRH3KMT2AKDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL1397993 0.82 HRH3 (0.56) HRH3KMT2AGPR119AKR1C3
SCHEMBL547046 0.82 CHRM2 (0.50) CHRM2CHRM1CHRM3GPR119KDM4E
SCHEMBL547045 0.82 CHRM2 (0.50) CHRM2CHRM1CHRM3GPR119KDM4E
SCHEMBL547468 0.80 CHRM2 (0.48) CHRM2CHRM1CHRM3GPR119KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118089-B1 INDOL-2-YL-PIPERAZIN-1-YL-METHANONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-05-12 EP disclosed